6
1
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4980 |
Betrixaban maleate
|
Factor Xa | Metabolism |
Betrixaban maleate 是一种非维生素 K 口服抗凝剂,其作用是由 Xa 因子的竞争性和可逆抑制作用驱动的。 | |||
T4341 |
Betrixaban
贝曲西班,PRT054021 |
Factor Xa | Metabolism |
Betrixaban (PRT054021) 是一种口服具有活力的选择性factor Xa(fXa) 抑制剂,IC50=1.5 nM。 | |||
T81204 |
SARS-CoV-2-IN-67
|
SARS-CoV | Microbiology/Virology |
SARS-CoV-2-IN-67 (Compound 16) 是抗SARS-CoV-2的维生素K衍生物,其在VeroE6/TMPRSS2细胞中EC50值为64.8 μM。该化合物能够抑制SARS-CoV-2 RdRp活性。 | |||
T81205 |
SARS-CoV-2-IN-66
|
SARS-CoV | Microbiology/Virology |
SARS-CoV-2-IN-66 (1),一种维生素K衍生物,作为SARS-CoV-2抑制剂,其在VeroE6/TMPRSS2细胞模型中的EC50值达到70.8 μM。 | |||
T37950 |
2-(Isopentylamino)naphthalene-1,4-dione
|
||
2-(Isopentylamino)naphthalene-1,4-dione is a vitamin K analog.1It inhibits spasms induced by pentylenetetrazole and tonic hindlimb extension induced by maximal electroshock (MES) in mice (ED50s = 349.2 and 108.1 mg/kg, respectively). It also protects mice against seizures in the 6 Hz psychomotor seizure test (ED50s = 152.7 and 263.7 mg/kg at stimulus intensities of 32 and 44 mA, respectively). 1.Li, X., Himes, R.A., Prosser, L.C., et al.Discovery of the first vitamin K analogue as a potential tr... | |||
T21693 |
PPM-18
|
||
PPM-18 (NSC 73233) 是一种有效的抗炎剂,可抑制一氧化氮合酶的表达。PPM-18 是有效的 iNOS 表达抑制剂,可阻断 NF-κB 与启动子的结合。PPM-18 是维生素 K 的类似物,通过 ROS 和 AMPK 信号通路诱导膀胱癌细胞自噬和凋亡。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2336 |
Vitamin K2
Menatetrenone,四烯甲萘醌 |
Endogenous Metabolite | Metabolism |
Vitamin K2 (Menatetrenone) 是内源性代谢产物的一种。 |