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Cat. No. Product Name Target Signaling Pathways
T6720 Vatalanib dihydrochloride

CGP-797870 dihydrochloride,ZK-222584 dihydrochloride,Vatalanib 2HCl,PTK787 dihydrochloride,Vatalanib (PTK787) 2HCl,CGP-79787 dihydrochloride,瓦他拉尼

Apoptosis; VEGFR; PDGFR Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
Vatalanib dihydrochloride (PTK787 dihydrochloride) 是一种VEGFR2/KDR 的抑制剂,其IC50值为37nM。
T17219 Vatalanib free base

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
Vatalanib free base 是一种 VEGFR2/KDR 的抑制剂,其IC50=37nM。
T71897 Vatalanib succinate

Vatalanib succinate is a VEGFR, PDGFR-β, c-Kit, c-Fms, and aromatase inhibitor.
T69888 SB02024

SB02024 is a VPS34 inhibitor. SB02024 activates cGAS-STING signaling and sensitizes tumors to STING agonist. SB02024 blocked autophagy in vitro and reduced xenograft growth of two breast cancer cell lines, MDA-MB-231 and MCF-7, in vivo. Vps34 inhibitor significantly potentiated cytotoxicity of Sunitinib and Erlotinib in MCF-7 and MDA-MB-231 in vitro in monolayer cultures and when grown as multicellular spheroids. Our data suggests that inhibition of autophagy significantly improves sensitivity...
T69487 ZK-261557

ZK-261557 is a new oral antiangiogenic molecule that inhibits all known vascular endothelial growth factor receptors. Vatalanib is under investigation for the treatment of solid tumors.

化合物

Vatalanib dihydrochloride
Cat.No: T6720
Synonym: CGP-797870 dihydrochloride,ZK-222584 dihydrochloride,Vatalanib 2HCl,PTK787 dihydrochloride,Vatalanib (PTK787) 2HCl,CGP-79787 dihydrochloride,瓦他拉尼
Target: Apoptosis, VEGFR, PDGFR
Vatalanib free base
Cat.No: T17219
Synonym:
Target: VEGFR
Vatalanib succinate
Cat.No: T71897
Synonym:
Target:
SB02024
Cat.No: T69888
Synonym:
Target:
ZK-261557
Cat.No: T69487
Synonym:
Target:
TargetMol Loading
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