Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13312L |
Seviteronel
VT-464 |
P450; Androgen Receptor | Endocrinology/Hormones; Metabolism |
Seviteronel (VT-464) 是一种新型 CYP17 裂解酶抑制剂和雄激素受体拮抗剂,可用于研究乳腺癌和前列腺癌。 | |||
T13313 |
Seviteronel racemate
VT-464 (racemate) |
Others | Others |
Seviteronel racemate is the racemate form of Seviteronel and is a potent inhibitor of CYP17 lyase. | |||
T13312 |
Seviteronel R enantiomer
VT-464 (R enantiomer) |
Others | Others |
Seviteronel R enantiomer is the R enantiomer of Seviteronel and is a potent inhibitor of CYP17 lyase (IC50: 69 nM for h-Lyase). |