Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T39717 |
VGSC blocker-1
|
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VGSC blocker-1 is a powerful small molecule that serves as a blocker for the neonatal isoform of the VGSC subtype known as Nav1.5 (nNav1.5). It effectively blocks INa peak currents by 34.9% at a concentration of 1 μM, and demonstrates a 0.3% inhibition of cell invasion at the same concentration in the MDA-MB-231 human breast cancer cell line, without compromising cell viability. | |||
T15260 |
Evenamide
NW-3509 |
Sodium Channel | Membrane transporter/Ion channel |
Evenamide (NW-3509) 是一种口服有效的电压门控钠通道 (sodium channel, VGSC) 阻滞剂,Ki 为 0.4 µM,在精神分裂症中有研究价值。Evenamide 在精神病,躁狂症,抑郁和攻击性的各种啮齿动物模型中具有显著功效。 | |||
T80626 |
VGSCs-IN-1
|
Sodium Channel | Membrane transporter/Ion channel |
VGSCs-IN-1 是一种有效的 VGSC 抑制剂,是一种 Riluzole 的 2-哌嗪类似物,在Nav1.4上展现出良好的阻断活性。VGSCs-IN-1可用于研究细胞兴奋性障碍。 | |||
T9751 |
Transfluthrin
|
Others | Others |
Transfluthrin 是一种挥发性拟除虫菊酯类杀虫剂,针对昆虫电压门控钠通道 (VGSC)。 | |||
T80427 |
Jingzhaotoxin-II
|
Sodium Channel | Membrane transporter/Ion channel |
Jingzhaotoxin-II是由32个氨基酸组成的神经毒素,包括两个酸性残基和两个碱性残基。该毒素能够抑制电压门控钠通道(VGSC),并在心肌细胞上明显减缓TTX抗性(TTX-R) VGSC的快速失活,其IC50值为0.26μM。 | |||
T80493 |
µ-Conotoxin BuIIIA
|
Sodium Channel | Membrane transporter/Ion channel |
μ-Conotoxin BuIIIA是从Cone snails毒液中提取的一种毒性肽类VGSC阻滞剂,常用于神经系统疾病的研究。 | |||
T80491 |
µ-Conotoxin BuIIIB
Mu-Conotoxin BuIIIB |
Sodium Channel | Membrane transporter/Ion channel |
μ-Conotoxin BuIIIB (Mu-Conotoxin BuIIIB) 是一种从Cone snails毒液中分离出的肽类分子,专门抑制哺乳动物神经元的电压门控钠通道 (VGSC),以用作研究离子通道功能的生物探针。它在神经系统疾病(例如疼痛)的研究中具有潜在应用价值。 | |||
T80159 |
µ-Conotoxin KIIIA
|
Sodium Channel | Membrane transporter/Ion channel |
μ-Conotoxin KIIIA,一种具有镇痛功能的μ-芋螺毒素,源自Conus kinoshitai。该化合物通过阻断哺乳动物神经元的电压门控钠通道(VGSC) (Nav1.2),可应用于疼痛研究领域。 |