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Cat. No. Product Name Target Signaling Pathways
T13237L Ropsacitinib

Tyk2-IN-8,PF-06826647

Tyrosine Kinases Tyrosine Kinase/Adaptors
Ropsacitinib (PF-06826647) 是一种选择性TYK2抑制剂。Ropsacitinib 与Tyk2催化活性JH1结构域结合(IC50:17nM)。
T13232 TyK2-IN-2

PDE Metabolism
TyK2-IN-2 is a selective inhibitor of TYK2 (IC50s: 7 nM, 0.1 μM, and 0.05 μM for TYK2 JH2, IL-23, and IFNα).
T13234 Tyk2-IN-5

Others Others
Tyk2-IN-5 is a selective and orally active inhibitor of Tyk2 JH2 (Ki: 0.086 nM for Tyk2 JH2; IC50: 25 nM for IFNα).
T13235 Tyk2-IN-7

Others Others
Tyk2-IN-7 is an inhibitor of TYK2 JH2, binds to the TYK2 JH2 domain (IC50: 0.00053 μM; Ki.app: 0.00007 μM).
T13237 Tyk2-IN-9

Others Others
Tyk2-IN-9 (化合物26),作为一种高选择性Tyk-2抑制剂,展现出对TYK2-JH2的IC50为0.076 nM,及对JAK1-JH2的IC50为1.8 nM,显示其在炎症或自身免疫性疾病研究中的应用前景。
T13233 Tyk2-IN-3

Tyrosine Kinases Tyrosine Kinase/Adaptors
Tyk2-IN-3 is an inhibitor of Tyk2 pseudokinase (IC50: 485 nM).
T61658 TYK2-IN-11

TYK2-IN-11 (Compound 5B) is a potent and selective inhibitor of Tyk-2, providing inhibition to TYK2-JH2 and JAK1-JH2 with IC50 values of 0.016 nM and 0.31 nM, respectively. This compound demonstrates potential for advancing research in the area of inflammatory and autoimmune diseases [1].

化合物

Ropsacitinib
Cat.No: T13237L
Synonym: Tyk2-IN-8,PF-06826647
Target: Tyrosine Kinases
TyK2-IN-2
Cat.No: T13232
Synonym:
Target: PDE
Tyk2-IN-5
Cat.No: T13234
Synonym:
Target: Others
Tyk2-IN-7
Cat.No: T13235
Synonym:
Target: Others
Tyk2-IN-9
Cat.No: T13237
Synonym:
Target: Others
Tyk2-IN-3
Cat.No: T13233
Synonym:
Target: Tyrosine Kinases
TYK2-IN-11
Cat.No: T61658
Synonym:
Target:
TargetMol Loading
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