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3

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T63105 Topotecan hydrochloride hydrate

Topotecan hydrochloride hydrate 是一种口服具有活力的拓扑异构酶 I (Topoisomerase I) 抑制剂,具有抗癌作用。Topotecan hydrochloride hydrate 能够将细胞周期阻滞在 G0/G1 和 S 期,并诱导细胞凋亡。
T73411 PV-1019

NSC 744039

PV-1019 (NSC 744039) 是一种有效的选择性 Chk2抑制剂,IC50值为 24 nM。PV-1019 抑制Topotecan 诱导的Chk2自磷酸化。PV-1019 抑制 IR 诱导的细胞凋亡。
T71908 NU1085

NU1085 is a potent poly(ADP-ribose) polymerase (PARP) inhibitors have been developed that potentiate the cytotoxicity of ionizing radiation and anticancer drugs. The biological effects of NU1085 [Ki = 6 nM], in combination with temozolomide (TM) or topotecan (TP) have been studied in 12 human tumor cell lines (lung, colon, ovary, and breast cancer). Cells were treated with increasing concentrations of TM or TP +/- NU1085 (10 microM) for 72 h.

化合物

Topotecan hydrochloride hydrate
Cat.No: T63105
Synonym:
Target:
PV-1019
Cat.No: T73411
Synonym: NSC 744039
Target:
NU1085
Cat.No: T71908
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T5784 Topotecan

NSC 609669,拓扑替康,SKF 104864A

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Topotecan (NSC-609669) 是一种拓扑异构酶 I 抑制剂,通过抑制 DNA 拓扑异构酶起抗肿瘤作用,可用于治疗卵巢癌。
T1174 Topotecan hydrochloride

SKF 104864A,SKFS 104864A,NSC609699,Nogitecan HCl,NSC 609669,盐酸拓扑替康,Topotecan HCl

Apoptosis; Topoisomerase; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair
Topotecan hydrochloride (NSC609699) 是一种具有抗癌活性的拓扑异构酶I 抑制剂。

天然产物

Topotecan
Cat.No: T5784
Synonym: NSC 609669,拓扑替康,SKF 104864A
Target: Topoisomerase, Autophagy
Topotecan hydrochloride
Cat.No: T1174
Synonym: SKF 104864A,SKFS 104864A,NSC609699,Nogitecan HCl,NSC 609669,盐酸拓扑替康,Topotecan HCl
Target: Apoptosis, Topoisomerase, Autophagy
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