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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T41248 |
Thiocolchicine
|
Microtubule Associated | Cytoskeletal Signaling |
Thiocolchicine 是一种有效的微管蛋白聚合抑制剂,IC50 为 2.5 µM,Ki 为 0.7 µM。 Thiocolchicine 诱导细胞凋亡。 Thiocolchicine 可用作 ADC 技术中的 ADC 细胞毒素。 | |||
T31000 |
Colchicine, N-deacetyl-10-thio-
N-Deacetylthiocolchicine,Desacetyl thiocolchicine,Deacetylthiocolchicine |
||
Colchicine, N-deacetyl-10-thio- is a biochemical. | |||
T31255 |
Deacetylthiocolchicine hydrochloride
Deacetylthiocolchicine chlorhydrate,Deacetylthiocolchicine HCl |
||
Deacetylthiocolchicine hydrochloride is a biochemical. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2S1464 |
Thiocolchicoside
硫秋水仙苷;噻可撒可,Thiocolchicine 2-glucoside analog,硫秋水仙苷,Coltramyl |
Others; GABA Receptor | Membrane transporter/Ion channel; Neuroscience; Others |
Thiocolchicoside (Thiocolchicine 2-glucoside analog) 是秋水仙碱的半合成硫衍生物,是竞争性 GABAA 受体拮抗剂和甘氨酸受体拮抗剂。它是肌肉松弛剂,具有抗炎作用,可用于缓解疼痛的研究。 |