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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7461 |
2,4-Diamino-6-hydroxypyrimidine
DAHP,2,4-二氨基-6-羟基嘧啶 |
Reactive Oxygen Species; NO Synthase | Immunology/Inflammation; Metabolism; NF-κB |
2,4-Diamino-6-hydroxypyrimidine (DAHP) 是GTP cyclohydrolase I(蛋白从头合成中的限速酶) 的选择性抑制剂。它能够抑制NO 的产生以及阻断 Tetrahydrobiopterin (BH4) 的合成。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T17056 |
Tetrahydrobiopterin
Sapropterin,BH4,(Rac)-Sapropterin |
NOS; Endogenous Metabolite | Immunology/Inflammation; Metabolism |
Tetrahydrobiopterin (BH4) 是芳香族氨基酸羟化酶的辅因子, 也是一氧化氮合酶 (NOS) 的必需辅因子,可用于研究如高血压、高胆固醇血症、糖尿病等内皮功能障碍。 | |||
T19160 |
7,8-Dihydro-L-biopterin
|
Endogenous Metabolite | Metabolism |
7,8-Dihydro-L-biopterin 是一种四氢生物蝶呤的氧化产物。 | |||
T38250 | L-Sepiapterin | ||
L-Sepiapterin, also known as Sepiapterin, is a precursor compound crucial for the production of tetrahydrobiopterin (BH4), which serves as a coenzyme for endothelial nitric oxide synthase (eNOS). This compound demonstrates its efficacy by improving endothelial dysfunction in small mesenteric arteries from db/db mice and promoting angiogenesis. Moreover, L-Sepiapterin exerts inhibitory effects on cellular proliferation and migration in ovarian cancer cells through the down-regulation of p70S6K-de... |