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抑制剂 & 化合物

5

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Cat. No. Product Name Target Signaling Pathways
T21508 Anhydrotetracycline hydrochloride

Antibacterial; Antibiotic Microbiology/Virology
Anhydrotetracycline hydrochloride 是四环素的生物合成前体,是广谱的、有效的竞争性四环素破坏酶抑制剂。它是真核细胞中四环素控制的基因表达系统的效应子。
T1101 Minocycline hydrochloride

Minocycline HCl,盐酸米诺环素,美满霉素

HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic Chromatin/Epigenetic; Metabolism; Microbiology/Virology
Minocycline hydrochloride (Minocycline HCl) 是四环素抗生素,具有出色的吸收和组织渗透性,可用于多种细菌感染以及痤疮的治疗。米诺环素可导致在开始治疗后 1 至 3 个月内发生的急性肝炎样综合征或通常在长期治疗后具有自身免疫特征的更隐匿的慢性肝炎。
T1140 Doxycycline hydrochloride

Doxylin,盐酸多西环素,Vibramycin,Hyclate

MMP; Antibacterial; Antibiotic Microbiology/Virology; Proteases/Proteasome
Doxycycline hydrochloride (Hyclate) 是一种四环素抗生素,是口服有效的广谱金属蛋白酶抑制剂,具有抗菌活性。

化合物

Anhydrotetracycline hydrochloride
Cat.No: T21508
Synonym:
Target: Antibacterial, Antibiotic
Minocycline hydrochloride
Cat.No: T1101
Synonym: Minocycline HCl,盐酸米诺环素,美满霉素
Target: HIF/HIF Prolyl-Hydroxylase, Antibacterial, Antibiotic
Doxycycline hydrochloride
Cat.No: T1140
Synonym: Doxylin,盐酸多西环素,Vibramycin,Hyclate
Target: MMP, Antibacterial, Antibiotic
Cat. No. Product Name Target Signaling Pathways
T0912 Tetracycline hydrochloride

NCI-c55561,盐酸四环素,Tetracycline HCl

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Tetracycline hydrochloride (NCI-c55561) 是一种广谱抗生素,抑制多种革兰氏阳性和革兰氏阴性细菌。
T21430 Oxytetracycline Hydrochloride

Biosolvomycin,盐酸土霉素,Oxytetracycline HCl,Oxytetracycline.HCl,Dalimycin,Oxytetracycline, Sodium Salt,Dalinmycin

Antiviral; Endogenous Metabolite; Antibacterial; HSV Immunology/Inflammation; Metabolism; Microbiology/Virology
Oxytetracycline Hydrochloride (Dalimycin) 是由 Streptomyces rimosus 生产的,一种具有抗菌活性的四环素衍生物。它干扰氨酰-tRNA 与 mRNA-核糖体复合物的结合,从而阻止肽延伸并抑制蛋白质合成。
T1400 Demeclocycline hydrochloride

地美环素,Declomycin,Clortetrin,盐酸地美环素,Detravis,Demeclocycline HCl

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Demeclocycline hydrochloride (Declomycin) 是四环素类抗生素,可治疗粉刺,莱姆病和支气管炎。
T1304 Chlortetracycline hydrochloride

Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Chlortetracycline hydrochloride (Isphamycin) 是一种特异性钙离子载体抗生素, 抑制氨酰 tRNA 结合到核糖体。
T0518 Methacycline hydrochloride

Rondomycin,盐酸甲烯土霉素,盐酸美他环素,Methacycline HCl

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Methacycline hydrochloride (Rondomycin) 是四环素抗生素,可抑制细菌蛋白质的合成。它是上皮-间质转化 (EMT) 抑制剂。它在体外可阻断 EMT,体内抑制纤维发生,不会直接影响 TGF-β1 Smad 信号传导。它是抗菌剂,有潜力研究肺纤维化。

天然产物

Tetracycline hydrochloride
Cat.No: T0912
Synonym: NCI-c55561,盐酸四环素,Tetracycline HCl
Target: ribosome, Antibacterial, Antibiotic
Oxytetracycline Hydrochloride
Cat.No: T21430
Synonym: Biosolvomycin,盐酸土霉素,Oxytetracycline HCl,Oxytetracycline.HCl,Dalimycin,Oxytetracycline, Sodium Salt,Dalinmycin
Target: Antiviral, Endogenous Metabolite, Antibacterial, HSV
Demeclocycline hydrochloride
Cat.No: T1400
Synonym: 地美环素,Declomycin,Clortetrin,盐酸地美环素,Detravis,Demeclocycline HCl
Target: ribosome, Antibacterial, Antibiotic
Chlortetracycline hydrochloride
Cat.No: T1304
Synonym: Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素
Target: ribosome, Antibacterial, Antibiotic
Methacycline hydrochloride
Cat.No: T0518
Synonym: Rondomycin,盐酸甲烯土霉素,盐酸美他环素,Methacycline HCl
Target: ribosome, Antibacterial, Antibiotic
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