Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13073L |
Taltobulin hydrochloride (228266-40-8 free base)
SPA-110 hydrochloride,Taltobulin hydrochloride,HTI-286 hydrochloride |
Others | Others |
Taltobulin hydrochloride is a synthetic analogue of the tripeptide hemiasterlin, is a potent agent of antimicrotubule that circumvents P-glycoprotein-mediated resistance in vitro and in vivo. | |||
TQ0141 |
Taltobulin
HTI-286,SPA-110 |
Apoptosis; Microtubule Associated | Apoptosis; Cytoskeletal Signaling |
Taltobulin (HTI-286) 是一种三肽半胱氨酸的合成类似物,是一种微管蛋白抑制剂,在体外抑制肝肿瘤细胞增殖和体内肿瘤生长。Taltobulin 具有细胞毒性,诱导有丝分裂停滞以及凋亡 (apoptosis),可用于研究乳腺癌和与微管组织相关的疾病。 | |||
T13073 |
Taltobulin trifluoroacetate
HTI-286 trifluoroacetate,SPA-110 trifluoroacetate |
Others | Others |
Taltobulin trifluoroacetate is a synthetic analogue of the tripeptide hemiasterlin, is a potent agent of antimicrotubule that circumvents P-glycoprotein-mediated resistance in vitro and in vivo. | |||
T75240 | Taltobulin hydrochloride | ||
Taltobulin hydrochloride (HTI-286 hydrochloride) 是一种合成的三肽半胱氨酸类似物,为高效抗微管剂,能够在体内外绕过P-糖蛋白介导的药物耐药性。该化合物通过抑制微管蛋白的聚合和破坏细胞内微管结构,进而引起细胞有丝分裂停滞和细胞凋亡。 |