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抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
TP1022 Protirelin Acetate

TSH-RF Acetate,TRH Acetate,TRF Acetate,醋酸普罗瑞林

Thyroid hormone receptor(THR); Endogenous Metabolite Endocrinology/Hormones; Metabolism
Protirelin Acetate (TRH Acetate) 是高度保守的神经肽,具有促甲状腺激素水平的激素控制作用,及神经调节的能力。
T6956L Protirelin Acetate(24305-27-9 free base)

Thyroliberin Acetate,TRF Acetate,Synthetic thyrotropin-releasing hormone Acetate,Lopremone Acetate,pGlu-His-Pro-NH2 Acetate,TRH Acetate

Thyroid hormone receptor(THR) Endocrinology/Hormones
Protirelin Acetate(24305-27-9 free base) (Thyroliberin Acetate) 是一种三肽,可刺激促甲状腺素和催乳素的释放。
T73825 TRFS-green

TRFS-green 是用于检测活细胞中、硫氧还蛋白还原酶 (TrxR)、且具有高度选择性的、off−on 荧光探针。TRFS-green 的 λmax 是 377 nm。
T75351 TP-TRFS

TP-TRFS 是高度选择性的一个硫氧还蛋白还原酶 (TrxR) 双光子荧光探针。
T34922 TRFS-red

TRFSred

TRFS-red is the first red emission off-on probe for thioredoxin reductase.
T33413 Mito-TRFS

MitoTRFS

Mito-TRFS is the first off-on probe for imaging the mitochondrial thioredoxin reductase (TrxR2) in live cells.
T10759 CEP-28122 mesylate salt (1022958-60-6 free base)

CEP-28122 mesylate salt

ALK Angiogenesis; Tyrosine Kinase/Adaptors
CEP-28122 mesylate salt (1022958-60-6 free base) 是一种高选择性的口服活性 ALK 抑制剂(在基于酶的 TRF 测定中,IC50:1.9 nM)。

化合物

Protirelin Acetate
Cat.No: TP1022
Synonym: TSH-RF Acetate,TRH Acetate,TRF Acetate,醋酸普罗瑞林
Target: Thyroid hormone receptor(THR), Endogenous Metabolite
Protirelin Acetate(24305-27-9 free base)
Cat.No: T6956L
Synonym: Thyroliberin Acetate,TRF Acetate,Synthetic thyrotropin-releasing hormone Acetate,Lopremone Acetate,pGlu-His-Pro-NH2 Acetate,TRH Acetate
Target: Thyroid hormone receptor(THR)
TRFS-green
Cat.No: T73825
Synonym:
Target:
TP-TRFS
Cat.No: T75351
Synonym:
Target:
TRFS-red
Cat.No: T34922
Synonym: TRFSred
Target:
Mito-TRFS
Cat.No: T33413
Synonym: MitoTRFS
Target:
CEP-28122 mesylate salt (1022958-60-6 free base)
Cat.No: T10759
Synonym: CEP-28122 mesylate salt
Target: ALK
Cat. No. Product Name Target Signaling Pathways
T6956 Protirelin

Lopremone,pGlu-His-Pro-NH2,Synthetic thyrotropin-releasing hormone,Thyroliberin,TRH,普罗瑞林,TRF

Thyroid hormone receptor(THR); Endogenous Metabolite Endocrinology/Hormones; Metabolism
Protirelin (Thyroliberin) 是高度保守的神经肽,具有促甲状腺激素水平的激素控制作用,及神经调节功能。

天然产物

Protirelin
Cat.No: T6956
Synonym: Lopremone,pGlu-His-Pro-NH2,Synthetic thyrotropin-releasing hormone,Thyroliberin,TRH,普罗瑞林,TRF
Target: Thyroid hormone receptor(THR), Endogenous Metabolite
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