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Cat. No.	Product Name	Target	Signaling Pathways
T34707	SST-02 SST 02,SST02
	SST-02 is a potent cationic lipid for siRNA-Lipid Nanoparticles. SST-02 possesses a simple chemical structure and is synthesized just in one step. SST-02 showed an ID50 of 0.02 mg/kg in the factor VII (FVII) model. Rats administered with 3 mg/kg of SST-02
TP2045	CH 275
	Potent somatostatin receptor 1 (sst1) agonist; displays selectivity for sst1 (IC50 values are 30.9 nM, 345 nM, > 1 μM, > 10 μM and > 10μM for human sst1, sst3, sst4, sst2 and sst5 respectively). Attenuates somatostatin release in the rat nucleus accumbens
T13004	SSTC3	Casein Kinase; Wnt/beta-catenin	Cytoskeletal Signaling; Metabolism; Stem Cells
	SSTC3 是一种酪蛋白激酶 1α (CK1α) 的激活剂，Kd 为 32 nM。SSTC3 具有潜在的抗肿瘤活性，可抑制 WNT 信号传导，抑制 SHH 髓母细胞瘤肿瘤的生长。
TP1370L	Crosstide TFA(171783-05-4 free base)	Others	Others
	Crosstide TFA(171783-05-4 free base) 是糖原合酶激酶 α/β 融合蛋白序列的肽类似物，是 Akt 的底物。
T76209	DSTYSLSSTLTLSK TFA
	DSTYSLSSTLTLSK TFA 是用于 Infliximab (Avakine) 定量检测的通用肽。Infliximab (Avakine) 是一种嵌合单克隆IgG1抗体，能特异性地结合到 TNF-α。
T64119	SSTR5 antagonist 2 hydrochloride
	SSTR5 antagonist 2 hydrochloride 是一种强效的、口服具有活力的、选择性的生长激素抑制激素(受体)亚型 5 (SSTR5) 拮抗剂，对 2 型糖尿病表现出研究潜力。
T13022	SSTR5 antagonist 2	Others	Others
	SSTR5 antagonist 2 is a highly potent, oral active and selective antagonist of somatostatin (receptor) subtype 5 (SSTR5),with potential to treat type 2 diabetes mellitus (T2DM).
TP1370	Crosstide
	Crosstide is a peptide analog of glycogen synthase kinase-3 (GSK-3) that functions as a natural substrate for Akt/PKB.
T83720	Biotin-Crosstide TFA Biotin-Gly-Arg-Pro-Arg-Thr-Ser-Ser-Phe-Ala-Glu-Gly-OH
	Biotin-crosstide是Akt底物crosstide的生物素化形式。
T76544	Cyclic SSTR agonist octreotide
	Cyclic SSTR agonist octreotide 是一种 Octreotide ，可作为生长抑素受体 (SSTR) 的激动剂。
T39191L	DSTYSLSSTLTLSK acetate DSTYSLSSTLTLSK acetate (177792-42-6 Free base)	Others	Others
	DSTYSLSSTLTLSK acetate 是可以用于英夫利昔单抗定量检测的人通用肽。
T80964	Toxic Shock Syndrome Toxin-1 (TSST-1) (58-78)
	Toxic Shock Syndrome Toxin-1 (TSST-1) (58-78)为T细胞增殖激活剂，以剂量依赖性方式增强人外周血单核细胞(PBMC)的体外增殖，适用于癌症与炎症免疫研究。
T13005	SSTR5 antagonist 1	Others	Others
	SSTR5 antagonist 1 is a selective, and orally available antagonist of somatostatin receptor subtype 5 (SSTR5)(IC50s of 9.6 and 57 nM for hSSTR5 and mSSTR5, respectively).
T39191	DSTYSLSSTLTLSK
	DSTYSLSSTLTLSK is a generic human peptide and can be used for infliximab quantitative detection. Infliximab (Avakine) is a chimeric monoclonal IgG1 antibody that specifically binds to TNF-α.
T60784	SSTR4 agonist 2
	SSTR4 agonist 2 是有效的生长抑素受体亚型 4 (SSTR4) 激动剂，在 SSTR4 相关的医学疾病研究中具有潜力。SSTR4 通路抑制痛觉和炎症。
T61130	SSTR4 agonist 3
	SSTR4 agonist 3 is a potent compound that activates the SSTR4 receptor. The SSTR4 receptor is highly expressed in the hippocampus and neocortex, which are regions associated with memory, learning, and Alzheimer's disease pathology. SSTR4 agonists demonstrate strong efficacy in rodent models of pain, both acute and chronic, by reducing peripheral nociception and inflammation. Considering its potential application in pain research, SSTR4 agonist 3 is of interest[1].
T60911	SSTR4 agonist 4
	SSTR4 agonist 4 是一种有效的SSTR4激动剂，具有用于疼痛研究的潜力。SSTR4 激动剂在与急性和慢性相关的抗外周伤害感受和抗炎活性相关疼痛的啮齿动物模型中有效。SSTR4 在海马和新皮质、记忆和学习区域以及阿尔茨海默病病理学中的表达水平相对较高。
T13022L	SSTR5 antagonist 2 TFA	Others	Others
	SSTR5 antagonist 2 TFA is a highly potent, oral active and selective antagonist of somatostatin (receptor) subtype 5 (SSTR5), with potential to treat type 2 diabetes mellitus (T2DM).
TP1570	Cortistatin-14	Somatostatin	GPCR/G Protein
	Cortistatin-14 是一种与生长抑素-14结构相似的神经肽，具有抗惊厥和神经保护作用，通过激活 sst（2）、生长素释放肽和 GABA（A/B）受体损害小鼠的识别记忆巩固，可用于研究脓毒症引发的认知障碍。
T76596	PRL 3195
	PRL 3195 是一种somatostatin receptor 拮抗剂，对人生长抑素受体 sst5、sst2、sst3、sst1和 sst4的Ki 分别为 6、17、66、1000 和 1000 nM。
T28220	NVP ACQ090 NVP-ACQ090,ACQ090,ACQ 090,NVPACQ090,ACQ-090
	NVP ACQ090 is a potent and subtype-selective somatostatin sst(3) receptor antagonist.
T75842	Cyclosomatostatin TFA
	Cyclosomatostatin TFA 作为一种有效的生长抑素(SST)受体拮抗剂，在直肠癌(CRC)细胞中通过抑制1型生长抑素受体(SSTR1)的信号传导，有效降低结细胞增殖、ALDH+细胞群体的大小以及球形成。
T76042	Angiopeptin TFA
	Angiopeptin TFA，一种生长抑素的环状八肽类似物，作为sst2/sst5受体部分激动剂，其IC50值为0.26 nM和6.92 nM。该化合物能够抑制生长激素释放及IGF-1(胰岛素样生长因子-1)的产生，同时抑制腺苷酸环化酶活性或刺激细胞外酸化。Angiopeptin TFA在冠状动脉粥样硬化的研究中显示出潜力。
T26225	SRA880 malonate SRA880,NVPSRA880,NVP-SRA880,NVP-SRA-880,NVP-SRA 880,NVP SRA880
	SRA880 is a non-peptide somatostatin sst(1) receptor antagonist which displays a significantly lower affinity for the other human recombinant somatostatin receptors ( pK(d)= 6.0) or a wide range of neurotransmitter receptors, except for the human dopamine
T82883	BIM-23027
	BIM-23027为高选择性sst2受体激动剂（EC50=0.32 nM），其功能效果类似生长抑素（SRIF，环状十四肽）。该化合物可促进多巴胺的释放，此过程通过Glu依赖的机制进行调控。
T35663	Cortistatin-29 (rat) (trifluoroacetate salt)
	Cortistatin-29 is a neuropeptide that is structurally similar to somatostatin-28. It is produced by cleavage of preprocortistatin to procortistatin, which is cleaved at dibasic amino acids to form cortistatin-29 and cortistatin-14 as well as other partial cleavage products. Cortistatin mRNA is expressed in the human brain and in interneurons of the rat hippocampus and cerebral cortex. Cortistatin-29 binds to somatostatin (SST) receptors with IC50 values of 2.8, 7.1, 0.2, 3, and 13.7 nM for SST1-...

化合物

Cat.No: T34707

Synonym: SST 02,SST02

Cat.No: TP2045

Cat.No: T13004

Target: Casein Kinase, Wnt/beta-catenin

Crosstide TFA(171783-05-4 free base)

Cat.No: TP1370L

Target: Others

DSTYSLSSTLTLSK TFA

Cat.No: T76209

SSTR5 antagonist 2 hydrochloride

Cat.No: T64119

SSTR5 antagonist 2

Cat.No: T13022

Target: Others

Cat.No: TP1370

Biotin-Crosstide TFA

Cat.No: T83720

Synonym: Biotin-Gly-Arg-Pro-Arg-Thr-Ser-Ser-Phe-Ala-Glu-Gly-OH

Cyclic SSTR agonist octreotide

Cat.No: T76544

DSTYSLSSTLTLSK acetate

Cat.No: T39191L

Synonym: DSTYSLSSTLTLSK acetate (177792-42-6 Free base)

Target: Others

Toxic Shock Syndrome Toxin-1 (TSST-1) (58-78)

Cat.No: T80964

SSTR5 antagonist 1

Cat.No: T13005

Target: Others

Cat.No: T39191

SSTR4 agonist 2

Cat.No: T60784

SSTR4 agonist 3

Cat.No: T61130

SSTR4 agonist 4

Cat.No: T60911

SSTR5 antagonist 2 TFA

Cat.No: T13022L

Target: Others

Cat.No: TP1570

Target: Somatostatin

Cat.No: T76596

Cat.No: T28220

Synonym: NVP-ACQ090,ACQ090,ACQ 090,NVPACQ090,ACQ-090

Cyclosomatostatin TFA

Cat.No: T75842

Angiopeptin TFA

Cat.No: T76042

SRA880 malonate

Cat.No: T26225

Synonym: SRA880,NVPSRA880,NVP-SRA880,NVP-SRA-880,NVP-SRA 880,NVP SRA880

Cat.No: T82883

Cortistatin-29 (rat) (trifluoroacetate salt)

Cat.No: T35663

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