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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T24865 |
Tenivastatin
L-654969,L654969,Simvastatin acid,L 654969,Simvastatin hydroxy acid |
ROS; HMG-CoA Reductase | Immunology/Inflammation; Metabolism |
Tenivastatin (Simvastatin acid) 是一种抗高脂血症的 HMG-CoA 还原酶抑制剂,抑制活性氧 (ROS) 产生,可用于研究原发性高脂血症。 | |||
T64292 | Simvastatin acid calcium hydrate | ||
Simvastatin acid (Tenivastatin) calcium hydrate 是一种具有口服具有活力的 HMG-CoA 还原酶 (HMGCR) 抑制剂。Simvastatin acid calcium hydrate 能够调节心肌细胞和转染 OATP3A1 基因的 HEK293 细胞的 OATP3A1 表达。Simvastatin acid calcium hydrate 也能够抑制吲哚酚硫酸盐 (indoxyl sulfate) 介导的活性氧 (ROS) 产生。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T16885 |
Simvastatin acid ammonium
辛伐他汀铵盐,Tenivastatin ammonium |
Others | Others |
Simvastatin ammonium is an active metabolite of simvastatin lactone mediated. Simvastatin ammonium reduces indoxyl sulfate-mediated reactive oxygen species and modulates OATP3A1 expression in cardiomyocytes and HEK293 cells transfected with the OATP3A1 ge |