Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0467 |
Sildenafil citrate
UK-92480 citrate,西地那非柠檬酸盐,枸橼酸西地那非 |
Apoptosis; PDE; Autophagy | Apoptosis; Autophagy; Metabolism |
Sildenafil citrate (UK-92480 citrate) 是一种磷酸二酯酶 5 抑制剂,IC50为 5.22 nM。 | |||
T36062 | N-Desmethyl Sildenafil (citrate) | ||
N-Desmethyl sildenafil is a major metabolite of sildenafil . N-Desmethyl sildenafil is formed via oxidative metabolism of sildenafil by the cytochrome (CYP) P450 isoforms CYP3A4, CYP3A5, and CYP3A7. |