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Cat. No. Product Name Target Signaling Pathways
T0272 Nilutamide

尼鲁米特,RU23908

Androgen Receptor Endocrinology/Hormones
Nilutamide (RU23908) 是一种非甾体抗雄激素药物,有用于转移性前列腺癌的潜力。
T12770 RR-11a analog

aza-peptide Michael acceptor, 7a

Parasite Microbiology/Virology
RR-11a analog (aza-peptide Michael acceptor, 7a) 是一种天冬酰胺酰内肽酶抑制剂,对阴道毛滴虫中的 AE1、蓖麻硬蜱中的 AE 和曼氏血吸虫中的 AE 的 IC50 分别为 4.5 nM、4.5 nM 和 31 nM。
T61549 HDAC8-IN-2

HDAC8-IN-2 (compound 5o) is a potent HDAC8 inhibitor, with IC50 values of 0.27 μM and 0.32 μM for smHDAC8 (Schistosoma mansoni histone deacetylase 8) and hHDAC8, respectively. It effectively kills schistosome larvae and greatly reduces egg laying in adult worm pairs [1].
T34809 Teroxalene hydrochloride

Teroxalene HCl,NSC 138704

Teroxalene Hydrochloride is disubstituted piperazine used to treat animals with Schistosoma mansoni.
T69421 Hydrolapachol

Hydrolapachol is a novel potent and selective inhibitor of schistosoma mansoni dihydroorotate dehydrogenase (smdhodh)
T33957 PF-Alkyne

PF Alkyne

PF-Alkyne is a fluorophosphonate-based probe which specifically and covalently reacts with the tyrosine-111 residue of the Schistosoma japonicum GST (sjGST) tag. PF-Alkyne rapidly and site-selectively immobilizes sjGST fusion proteins.
T61538 Antiparasitic agent-10

Antiparasitic agent-10 (Compound 94) is a potent anti-parasitic agent specifically designed to target and combat parasitic infections. It demonstrates notable anti-schistosomal activity, particularly against adults of Schistosoma mansoni. As a result, this compound holds significant potential for utilization in Schistosomiasis research as a viable treatment option [1].
T78391 DAUDA

DAUDA (11-(dansylamino) undecanoic acid)是一种荧光脂肪酸类似物,对环境变化敏感。该分子通过调整其发射强度和荧光光谱与结合蛋白发生相互作用。在研究中,DAUDA用于评估天然脂肪酸与曼氏血吸虫Sm14脂肪酸结合蛋白多晶型的相对亲和力。
T78619 Z-Pro-Pro-CHO

Prolyl Endopeptidase (PREP) Metabolism; Proteases/Proteasome
Z-Pro-Pro-CHO为一种有效的脯氨酰寡肽酶抑制剂,其具有针对人类及曼氏血吸虫脯氨酰寡肽酶的较低半抑制浓度(IC50),分别为0.16 μM和0.01 μM。

化合物

Nilutamide
Cat.No: T0272
Synonym: 尼鲁米特,RU23908
Target: Androgen Receptor
RR-11a analog
Cat.No: T12770
Synonym: aza-peptide Michael acceptor, 7a
Target: Parasite
HDAC8-IN-2
Cat.No: T61549
Synonym:
Target:
Teroxalene hydrochloride
Cat.No: T34809
Synonym: Teroxalene HCl,NSC 138704
Target:
Hydrolapachol
Cat.No: T69421
Synonym:
Target:
PF-Alkyne
Cat.No: T33957
Synonym: PF Alkyne
Target:
Antiparasitic agent-10
Cat.No: T61538
Synonym:
Target:
DAUDA
Cat.No: T78391
Synonym:
Target:
Z-Pro-Pro-CHO
Cat.No: T78619
Synonym:
Target: Prolyl Endopeptidase (PREP)
TargetMol Loading
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