Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1520 |
Aliskiren hemifumarate
阿利克仑半富马酸盐,CGP 60536,SPP 100,CGP60536B |
RAAS; Autophagy | Autophagy; Endocrinology/Hormones |
Aliskiren hemifumarate (CGP60536B) 一种可口服非肽肾素抑制剂,IC50为1.5 nM,具有抗高血压活性。 | |||
T72526 |
Aliskiren fumarate
CGP 60536 fumarate,SPP 100 fumarate,CGP 60536 fumarate ; CGP60536B fumarate ; SPP 100 fumarate,CGP60536B fumarate |
||
Aliskiren fumarate是一种口服有效、选择性的肾素(renin)抑制剂,IC50值为1.5 nM。适用于高血压、心血管疾病和癌症恶病质的研究。 | |||
T19187 |
Aliskiren D6 hemifumarate
CGP 60536 D6 hemifumarate,SPP 100 D6 hemifumarate,CGP60536B D6 hemifumarate |
RAAS | Endocrinology/Hormones |
Aliskiren (CGP 60536) D6 hemifumarate is a deuterium-labeled Aliskiren hemifumarate. Aliskiren hemifumarate is a direct and orally active renin inhibitor (IC50: 1.5 nM). | |||
T10282 |
Aliskiren D6 Hydrochloride
SPP 100 D6 Hydrochloride,CGP60536B D6 Hydrochloride,CGP 60536 D6 Hydrochloride |
Others | Others |
Aliskiren (CGP 60536) D6 Hydrochloride is a deuterium-labeled Aliskiren. Aliskiren hemifumarate is a direct and orally active renin inhibitor (IC50: 1.5 nM). | |||
T27300 |
Olorofim
Olorofim,F901318,F-901318 |
||
Olorofim 是一种新型的选择性抗真菌化合物,对烟曲霉DHODH 具有抑制作用(IC50:44 nM),对人类DHODH 几乎没有抑制作用(>100 uM)。Olorofim 对青霉菌属、皮炎杆菌属、镰刀菌属等各种致病性丝状和二形真菌有很好的疗效。 | |||
T64163 | Aliskiren hydrochloride | ||
Aliskiren (CGP 60536; CGP60536B; SPP 100) hydrochloride 是一种选择性的、口服具有活力的、肾素 (renin) 抑制剂 (IC50: 1.5 nM)。Aliskiren hydrochloride 能够用于研究高血压、心血管疾病和癌症恶病质。 |