Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T69877 |
SPOP-IN-6lc
|
Apoptosis | Apoptosis |
SPOP-IN-6lc 是一种有效的 SPOP 抑制剂,在癌症中有多种作用,在多种肿瘤中有抑癌作用,在肾癌中却发挥着癌基因功能。SPOP-IN-6lc 可用于研究细胞信号传送和细胞凋亡。 | |||
T16922 |
SPOP-IN-6b
2-Imino-10-methyl-N-(3-morpholinopropyl)-5-oxo-1-phenethyl-1,5-dihydro-2H-dipyrido[1,2-a:2',3'-d]pyrimidine-3-carboxamide |
Others | Others |
SPOP-IN-6b 是一种有效的斑点型 POZ 蛋白 (SPOP) 抑制剂,IC50 为 3.58 μM,可用于肾癌治疗的研究。 | |||
T39593 |
SPOP-IN-6b hydrochloride
|
||
SPOP-IN-6b hydrochloride is a highly effective inhibitor of speckle-type POZ protein (SPOP), exhibiting an IC50 value of 3.58 μM. | |||
T64055 | SPOP-IN-6b dihydrochloride | ||
SPOP-IN-6b dihydrochloride 是斑型 POZ 蛋白 (SPOP) 的有效抑制剂 (IC50: 3.58 μM)。 | |||
T8658 |
NEO2734
EP31670 |
Epigenetic Reader Domain; Histone Acetyltransferase | Chromatin/Epigenetic |
NEO2734 (EP31670) 是一种具有口服活性的选择性 p300/CBP 和 BET 溴结构域抑制剂,其 IC50值均小于30 nM,可用于前列腺癌的研究。 |