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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T70953 AZ5576 racemate

AZ5576 racemate is a racemic mixture of AZ5576 isomers. AZ5576 is a potent, highly selective, and orally bioavailable inhibitor of Cdk9 that inhibits Cdk9 enzyme activity with an IC50 <5nM and decreases phosphorlyation of Ser2-RNAPII in cells with an IC50 of 96nM. In the MLL-fusion containing acute myeloid leukemia (AML) line, MV411, short-term treatment with AZ5576 led to a rapid dose-dependent decrease in pSer2-RNAPII with concomitant loss of Mcl1 mRNA and protein, resulting in the cleavage a...
T60152 AZ5576

CDK Cell Cycle/Checkpoint
AZ5576 是一种有效且高选择性的 CDK9抑制剂。AZ5576 可用于血液恶性肿瘤研究。

化合物

AZ5576 racemate
Cat.No: T70953
Synonym:
Target:
AZ5576
Cat.No: T60152
Synonym:
Target: CDK
Cat. No. Product Name Target Signaling Pathways
T70955 Vinaxanthone

SM-345431

Phospholipase; Antibacterial Metabolism; Microbiology/Virology
Vinaxanthone (SM-345431) 是一种从青霉菌中提取的小分子化合物,是一种具有选择性和有效性的 semaphorin3A、phospholipase C (PLC) 和 FabI 抑制剂,抑制semaphorin3A 和 FabI。Vinaxanthone 具有抗菌活性,阻止细胞内脂肪酸合成,抑制金黄色葡萄球菌的生长。

天然产物

Vinaxanthone
Cat.No: T70955
Synonym: SM-345431
Target: Phospholipase, Antibacterial
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