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Cat. No. Product Name Target Signaling Pathways
T12928 SK33

Androgen Receptor Endocrinology/Hormones
SK33 是一种有效的组织选择性抗雄激素药物,是一种肌醇类似物,能够降低雄激素受体 (AR) 的转录活性。
T5745 GSK3326595

EPZ015938

Histone Methyltransferase Chromatin/Epigenetic
GSK3326595 (EPZ015938) 是一种选择性可逆的蛋白精氨酸甲基转移酶 5 抑制剂,IC50为6.2 nM,具有广谱的抗增殖活性。
T11500L GSK3368715 dihydrochloride

EPZ019997 dihydrochloride,GSK3368715 2HCl,EPZ019997 2HCl

Histone Methyltransferase Chromatin/Epigenetic
GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) 是一种具有口服活性和高效性的 I 型蛋白精氨酸甲基转移酶 (PRMTs) 抑制剂 ,具有抗癌和抗肿瘤活性,抑制PRMT1,PRMT3,PRMT4,PRMT6,PRMT8的活性,可用于研究晚期实体肿瘤。
T22342 GSK3368715 3HCl

EPZ019997 3HCl,GSK3368715(EPZ019997)

Histone Methyltransferase Chromatin/Epigenetic
GSK3368715, a potent inhibitor of type I protein arginine methyltransferases (PRMT), could inhibit PRMT1, 3, 4, 6 and 8 with Kiapp vaules ranging from 1.5 to 81 nM.
T15439 GSK3395879

TRP/TRPV Channel Membrane transporter/Ion channel
GSK3395879 is a selective and orally bioavailable antagonist of transient receptor potential vanilloid-4 (TRPV4) (IC50: 1 nM for hTRPV4).
T11500 GSK3368715

EPZ019997

Histone Methyltransferase Chromatin/Epigenetic
GSK3368715 is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50s: 3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8)). It has strong anti-cancer activity.
T27473 GSK334429

GSK-334429,GSK 334429

GSK334429 is an antagonist of histamine H3 receptor.

化合物

SK33
Cat.No: T12928
Synonym:
Target: Androgen Receptor
GSK3326595
Cat.No: T5745
Synonym: EPZ015938
Target: Histone Methyltransferase
GSK3368715 dihydrochloride
Cat.No: T11500L
Synonym: EPZ019997 dihydrochloride,GSK3368715 2HCl,EPZ019997 2HCl
Target: Histone Methyltransferase
GSK3368715 3HCl
Cat.No: T22342
Synonym: EPZ019997 3HCl,GSK3368715(EPZ019997)
Target: Histone Methyltransferase
GSK3395879
Cat.No: T15439
Synonym:
Target: TRP/TRPV Channel
GSK3368715
Cat.No: T11500
Synonym: EPZ019997
Target: Histone Methyltransferase
GSK334429
Cat.No: T27473
Synonym: GSK-334429,GSK 334429
Target:
TargetMol Loading
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