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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T80130 |
SDF-1α (human)
|
CXCR | Autophagy; GPCR/G Protein; Immunology/Inflammation |
SDF-1α (human) 是一种能够与CXCR4受体相结合的单核细胞趋化剂,它在心肌梗死模型中的干细胞归巢、维持、生存、增殖、心肌细胞修复、血管形成以及心室重构过程扮演关键角色。SDF-1α (human) 常用于心血管病研究。 | |||
T76327 |
CTCE-0214
|
||
CTCE-0214 是一种 CXCR4(chemokine CXC receptor 4) 激动剂,是 SDF-1α 肽类似物。CTCE-0214 具有抗炎活性,可用于炎症败血症和系统性炎症综合征的研究。 | |||
T39787 |
KRH-3955 hydrochloride
|
||
KRH-3955 hydrochloride is a CXCR4 antagonist with oral bioavailability. It effectively inhibits the binding of SDF-1α to CXCR4, exhibiting an IC 50 of 0.61 nM. Additionally, KRH-3955 hydrochloride displays high potency and selectivity as an inhibitor of X4 HIV-1, with an EC 50 ranging from 0.3 to 1.0 nM. | |||
T63661 |
HF51116
|
||
HF51116 是 XCR4 的有效拮抗剂。HF51116 能够显著拮抗 SDF-1α 诱导的细胞迁移、钙动员和 CXCR4 内化,并利用 CXCR4 抑制 HIV-1 感染。HF51116 对HIV-1感染、造血干细胞动员和癌症转移表现出研究潜力。 | |||
T33267 |
Me6TREN 4HCl
Me6TREN Tetrahydrochloride,Me6-TREN Tetrahydrochloride,Me6 4HCl,Me 6 4HCl,Me-6 4HCl |
||
Me6TREN 4HCl is a potent and efficacious mobilizing agent of hematopoietic stem and progenitor cells (HSPCs) that can act by activating MMP-9 expression and disrupting the SDF-1α/CXCR4 axis, exhibiting more significant mobilizing effects than G-CSF or AMD | |||
T15805 |
LY2510924
|
Others | Others |
LY2510924 is an effective and selective CXCR4 antagonist. It blocks SDF-1 binding to CXCR4 (IC50: 0.079 nM). |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T9218 |
Andrograpanin
19-HYDROXY-8(17),13-LABDADIEN-16,15-OLIDE,新穿心莲内酯苷元 |
p38 MAPK | MAPK |
Andrograpanin (19-HYDROXY-8(17),13-LABDADIEN-16,15-OLIDE) 是来自穿心莲的一种天然产物,具有抗炎和抗感染活性。 |