Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T60962 |
SARS-CoV-2-IN-18
|
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SARS-CoV-2-IN-18 (Compound 26) 是 SARS-CoV-2 3C-样蛋白酶的有效抑制剂 (IC50 = 45 nM)。 | |||
T79661 |
SARS-CoV-2 3CLpro-IN-18
|
SARS-CoV | Microbiology/Virology |
SARS-CoV-2 3CLpro-IN-18(Compound 3C)为一种共价SARS-CoV-2 3CLpro抑制剂,具有0.478 μM的IC50值。在Vero E6细胞中对SARS-CoV-2展现出2.499 μM的EC50抑制活性,并显示出较低的细胞毒性(CC50> 200 μM)。 | |||
T79677 |
SARS-CoV-2-IN-58
|
Virus Protease | Microbiology/Virology |
SARS-CoV-2-IN-58(Compound 21H)是一种针对SARS-CoV-2Mpro的抗病毒剂,具有EC50值为18 μM和IC50值为0.35 μM的抑制活性。 |