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Cat. No. Product Name Target Signaling Pathways
T69358 S101

S101 is an inhibitor of proliferating T-cells, rescuing mice from superantigen-induced shock.
T3516 EDO-S101

Tinostamustine,Minomustine

HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair
EDO-S101 (Tinostamustine) 是一种泛 HDAC 抑制剂,IC50为 6 nM,对 HDAC1、HDAC2 和 HDAC3 的 IC50 值分别为 9、9 和 25 nM。
T70189 Navoximod phosphate

Navoximod phosphate is an indoleamine 2,3-dioxygenase (IDO) inhibitor, immunomodulator and antineoplastic.
T5170 KHS101 hydrochloride

盐酸KHS101

FGFR; Microtubule Associated Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
KHS101 hydrochloride 能够选择性的诱导神经元分化表型,能够与转化酸性含螺旋蛋白发生相互作用。
T15715 LAS101057

Adenosine Receptor GPCR/G Protein; Neuroscience
LAS101057 是一种新型可口服且具有有效性和选择性的 A2B receptor 拮抗剂,可用于研究哮喘。
T70190 Tinostamustine HCl

Tinostamustine, also known as EDO-S101, is an alkylatlng histone-deacetylase inhibitor (HDACi) fusion molecule. EDO-S101 is a functional pan-histone-deacetylase inhibitor and is assumed to potentiate the alkylating activity of the compound and/or may help to overcome resistance to other therapeutic agents.

化合物

S101
Cat.No: T69358
Synonym:
Target:
EDO-S101
Cat.No: T3516
Synonym: Tinostamustine,Minomustine
Target: HDAC
Navoximod phosphate
Cat.No: T70189
Synonym:
Target:
KHS101 hydrochloride
Cat.No: T5170
Synonym: 盐酸KHS101
Target: FGFR, Microtubule Associated
LAS101057
Cat.No: T15715
Synonym:
Target: Adenosine Receptor
Tinostamustine HCl
Cat.No: T70190
Synonym:
Target:
TargetMol Loading
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