Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11662L |
INT-777
S-EMCA |
GPCR19 | GPCR/G Protein |
INT-777(S-EMCA)是有效的 TGR5 激动剂,EC50 为 0.82 μM。 INT-777(S-EMCA)在大鼠蛛网膜下腔出血后通过 TGR3/cAMP/PKA 信号通路抑制 NLRP5-ASC 炎症小体介导的神经炎症。 | |||
T11662 |
INT-777 R-enantiomer
S-EMCA R enantiomer |
Others | Others |
INT-777 is the R-enantiomer of INT-777, less potent than INT-777,EC50 of 4.79 μM for TGR5. |