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Cat. No. Product Name Target Signaling Pathways
T1184 Rivaroxaban

BAY 59-7939,利伐沙班

Factor Xa; Thrombin Metabolism; Proteases/Proteasome
Rivaroxaban (BAY 59-7939) 是高效选择性的凝血因子 Xa (FXa) 直接抑制剂,IC50=0.7 nM,Ki 为 0.4 nM。
T67853 Rivaroxaban Impurity

Rivaroxaban-10

Factor Xa Metabolism
Rivaroxaban Impurity (Rivaroxaban-10) 是一种强效凝血因子Xa 抑制剂,IC50=66 nM。
T10174 5-R-Rivaroxaban

Factor Xa Metabolism
5-R-Rivaroxaban 是一种 Rivaroxaban 的 R 型对映体。其中 Rivaroxaban 是选择性的Factor Xa(FXa) 抑制剂。
T78215 Dechloro Rivaroxaban

Factor Xa; Others Metabolism; Others
Dechloro Rivaroxaban 是一种具有口服活性和高选择性的 Factor Xa 抑制剂。Dechloro Rivaroxaban 对人体内游离 FXa 的抑制作用显著。Dechloro Rivaroxaban 对凝血酶原以及纤维蛋白相关的 FXa 活性也有抑制效果。
T12736 Rivaroxaban-d4

BAY 59-7939 D4

Factor Xa Metabolism
Rivaroxaban D4 is a deuterium labeled Rivaroxaban. Rivaroxaban is a highly potent,selective and direct inhibitor of Factor Xa (FXa)(IC50:0.7 nM; Ki:0.4 nM).
T71096 GCC-4401C methanesulfonate

GCC-4401C methanesulfonate is a factor Xa inhibitor similar to rivaroxaban that is currently under development for venous thromboembolic disease (VTE).
T71362 GCC-4401C free base

GCC-4401C free base is a factor Xa inhibitor similar to rivaroxaban that is currently under development for venous thromboembolic disease (VTE).

化合物

Rivaroxaban
Cat.No: T1184
Synonym: BAY 59-7939,利伐沙班
Target: Factor Xa, Thrombin
Rivaroxaban Impurity
Cat.No: T67853
Synonym: Rivaroxaban-10
Target: Factor Xa
5-R-Rivaroxaban
Cat.No: T10174
Synonym:
Target: Factor Xa
Dechloro Rivaroxaban
Cat.No: T78215
Synonym:
Target: Factor Xa, Others
Rivaroxaban-d4
Cat.No: T12736
Synonym: BAY 59-7939 D4
Target: Factor Xa
GCC-4401C methanesulfonate
Cat.No: T71096
Synonym:
Target:
GCC-4401C free base
Cat.No: T71362
Synonym:
Target:
TargetMol Loading
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