Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12797 |
RU-SKI 43
RUSKI 43 |
Hedgehog/Smoothened; Acyltransferase | GPCR/G Protein; Metabolism; Stem Cells |
RU-SKI 43 是一种有效的选择性刺猬酰基转移酶 (Hhat) 抑制剂,IC50 为 850 nM。RU-SKI 43 具有抗癌活性,是治疗肺腺癌的潜在化合物。RU-SKI 43 通过独立于平滑化的非规范信号传导降低 Gli-1 激活,并抑制 Akt 和 mTOR 通路活性。 | |||
T12797L |
RU-SKI 43 hydrochloride
|
Others | Others |
RU-SKI 43 hydrochloride is a potent and selective inhibitor of Hedgehog acyltransferase (Hhat)(IC50 of 850 nM), has anti-cancer activity. |