Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T17227 |
Vernakalant Hydrochloride
RSD1235 hydrochloride |
Potassium Channel; Sodium Channel | Membrane transporter/Ion channel |
Vernakalant Hydrochloride (RSD1235 hydrochloride) 是一种混合电压和频率依赖性的 Na+ 和 K+ 通道阻断剂。Vernakalant 抑制 Kv1.5 channelwt,Kv1.5 channelI508F,Kv1.5 channelT479A,IC50 分别为 13.35±0.93 μM。 | |||
TQ0307 |
Vernakalant
RSD1235,维那卡兰 |
Potassium Channel | Membrane transporter/Ion channel |
Vernakalant (RSD-1235) is a mixed ion channel blocker. |