Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2282 |
RPI-1
|
Others; Phospholipase; c-Met/HGFR; c-RET | Apoptosis; Metabolism; Others; Tyrosine Kinase/Adaptors |
RPI1 是特异性的、口服具有活力的 2-吲哚啉酮Ret 酪氨酸激酶抑制剂,具有抗肿瘤作用。它能够抑制人甲状腺髓样癌 TT 细胞增殖、Ret 酪氨酸磷酸化、Ret 蛋白表达及 PLCgamma、ERKs 和 AKT 的活化。 | |||
T24737 |
Rpi 856 A
Rpi856 A,Rpi 856 B,Rpi-856 A,Rpi-856 B,Rpi856 B |
||
Rpi 856 A is a retrovirus protease inhibitor. It is effective against HIV-1 and HTLV-1 proteases. | |||
T26128 |
Rpi 856 C
Rpi-856 C,Rpi856 C,Rpi-856 D,Rpi856 D,Rpi 856 D |
||
Rpi 856 C is a retrovirus protease inhibitor from Streptomyces that is effective against HIV-1 and HTLV-1 proteases. |