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抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T79077 ROCK-IN-6

ROCK Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
ROCK-IN-6为一有效的ROCK2抑制剂,其IC50值为2.19 nM。该化合物具备用于研究青光眼及视网膜疾病的潜力。
T79832 ROCK2-IN-6

ROCK Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
ROCK2-IN-6 (Comp A) 是一種选择性针对ROCK2的抑制剂,适用于研究ROCK介导的病症、自身免疫性疾病以及炎症。
T78205 ROCK2-IN-6 hydrochloride

ROCK Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
ROCK2-IN-6 hydrochloride (Comp A)为一种选择性ROCK2抑制剂,适用于研究ROCK介导的疾病、自身免疫性病症与炎症。
T37847 Zonisamide-13C2,15N

Zonisamide-13C2,15N

Zonisamide-13C2,15N is intended for use as an internal standard for the quantification of zonisamide by GC- or LC-MS. Zonisamide is an antiepileptic agent.1 It selectively inhibits the repeated firing of sodium channels (IC50 = 2 μg/ml) in mouse embryo spinal cord neurons and inhibits spontaneous channel firing when used at concentrations greater than 10 μg/ml.2 In rat cerebral cortex neurons, zonisamide (1-1,000 μM) inhibits T-type calcium channels with a maximum reduction of 60% of the calcium...

化合物

ROCK-IN-6
Cat.No: T79077
Synonym:
Target: ROCK
ROCK2-IN-6
Cat.No: T79832
Synonym:
Target: ROCK
ROCK2-IN-6 hydrochloride
Cat.No: T78205
Synonym:
Target: ROCK
Zonisamide-13C2,15N
Cat.No: T37847
Synonym: Zonisamide-13C2,15N
Target:
Cat. No. Product Name Target Signaling Pathways
T4S1962 beta-Asarone

β-细辛脑,(Z)-1,2,4-三甲氧基-5-丙烯基苯;顺式细辛脑,Cis-Isoasarone,Cis-Asarone,Cis-Isoelemicin

NF-κB; JNK MAPK; NF-κB
beta-Asarone (Cis-Isoelemicin) 是一种石菖蒲中的主要成分,具有免疫抑制、促进安定、中枢神经系统抑制、降温等功能。它可透过血脑屏障,能够预防帕金森病。

天然产物

beta-Asarone
Cat.No: T4S1962
Synonym: β-细辛脑,(Z)-1,2,4-三甲氧基-5-丙烯基苯;顺式细辛脑,Cis-Isoasarone,Cis-Asarone,Cis-Isoelemicin
Target: NF-κB, JNK
TargetMol Loading
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