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Cat. No. Product Name Target Signaling Pathways
T5513 RO-3

P2X Receptor Membrane transporter/Ion channel; Neuroscience
RO3 是一种能透过大脑的P2X3和P2X2/3拮抗剂,口服有活性。它对人同型多聚体 P2X3和异型多聚体 P2X2/3受体的 pIC50分别为 5.9 和 7.0。
T30611 Bufuralol

Ro3-4787,Ro 3-4787,Ro-3-4787

Bufuralol is a Adrenergic Agent.
TP2206 [Leu31,Pro34]-Neuropeptide Y (porcine)

LEU 31, PRO34]-神经肽Y(猪)

Neuropeptide Y Receptor GPCR/G Protein; Neuroscience
[Leu31,Pro34]- Neuropeptide Y (porcine) 是神经肽 Y (NPY) 的一种类似物,是对NPY Y1受体有选择性的激动作用。它表现出抗焦虑作用。
TP2020L [Pro3]-GIP (Mouse) acetate

Others Others
[Pro3]-GIP (Mouse) acetate 是鼠源[Pro3]-GIP。[Pro3]-GIP 是一种 GIP receptor 拮抗剂。
T69360 RO3244794

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
RO3244794是一种具有选择性的前列环素 (IP)受体拮抗剂,可用于研究肝脏损伤。
T2634 Ro3280

RO 3280,Ro5203280

PLK Cell Cycle/Checkpoint
Ro3280 (Ro5203280) 是一种高度选择性的PLK1抑制剂,IC50和Kd 值分别为 3 nM 和 0.09 nM。
T76313 (Pro3) GIP, human

(Pro3) GIP, human ((Pro3)Gastric Inhibitory Peptide, human) 是一种有效、稳定和特异性的人 GIP 受体完全激动剂。(Pro3) GIP, human 对人 GIPR 具有高结合亲和力,Ki/ Kd 值为 0.90 nM。(Pro3) GIP, human 可用于肥胖相关糖尿病的研究。
T76441 (Pro34)-Peptide YY (human)

(Pro34)-Peptide YY (human) 是 Peptide YY/neuropeptide Y 受体的高度 Y1选择性全激动剂。
T34370 RO320-2947/001

RO-320-2947/001,RO 320-2947/001

RO320-2947/001 is a bioactive chemical.
TP2021 [Pro3]-GIP (Rat)

High affinity rat GIP receptor partial agonist (Kd = 13 nM). Increases cAMP accumulation in COS-7 cells transfected with rat GIP receptor, while also acting as a competitive antagonist of GIP.
T75912 [Leu31,Pro34]-Neuropeptide Y(human,rat) TFA

[Leu31,Pro34]-Neuropeptide Y(human,rat) TFA 是一种针对神经肽 YY1受体的特定激动剂,并亦能够激活Y4和Y5受体。该化合物能提高麻醉大鼠的血压并增加食物摄入。
TP1985 [Leu31,Pro34]-Neuropeptide Y(human,rat)

[Leu31,Pro34]-Neuropeptide Y (human, rat)

High affinity neuropeptide Y Y1 receptor agonist (Ki = 0.39 nM). Also shows affinity for Y4 and Y5 receptors.
TP2020 [Pro3]-GIP (Mouse)

GIP receptor antagonist (IC50 = 2.6μM). Inhibits GIP-stimulated insulin release from pancreatic β cells in vitro. In ob/ob mice, blocks the effects of GIP on insulin release and plasma glucose levels. Also improves intraperitoneal glucose tolerance, insul
T34903 TO-PRO3 iodide

TOPRO3 iodide,TO-PRO3 iodide salt

TO-PRO3 iodide is a nucleic acid stain that can stain the nucleus of cells in different states, including living, early apoptotic, and necrotic cells.
T71420 RO314724

RO314724 is a HDAC inhibitor. RO314724 is also a a reversible, tightly binding, MMP inhibitor with a Ki of 26 nm. Matrix metalloproteinases (MMPs) belong to the key enzymes of the proteolytic destruction of cartilage matrix during chronic rheumatic diseases. Ro314724 displayed MMP-proteoglycanase inhibitory activity both in vitro and ex vivo and proved to be not harmful to the morphology, viability and proteoglycan biosynthesis of bovine articular cartilage explants.
T83499 [D-Phe2,6, Pro3]-LH-RH

[D-Phe2,6, Pro3]-LH-RH是一种促黄体生成素释放激素(LHRH)的高效拮抗剂,具有特定氨基酸序列变异。
T80087 (Leu31,Pro34)-Peptide YY (human) (TFA)

Neuropeptide Y Receptor GPCR/G Protein; Neuroscience
'(Leu31,Pro34)-Peptide YY (human)(TFA)' 为 '(Leu31,Pro34)-Peptide YY (human)' 的 TFA 盐形式,该化合物为 Peptide YY 的衍生物,兼具高效和选择性的 Y1 受体激动剂特性,其 KD 值为 1.0 nM。
T76442 (Leu31,Pro34)-Peptide YY (human)

(Leu31,Pro34)-Peptide YY (human) 是一种 Peptide YY 的衍生物,是一种有效的、选择性的 Y1激动剂,KD 为 1.0 nM。

化合物

RO-3
Cat.No: T5513
Synonym:
Target: P2X Receptor
Bufuralol
Cat.No: T30611
Synonym: Ro3-4787,Ro 3-4787,Ro-3-4787
Target:
[Leu31,Pro34]-Neuropeptide Y (porcine)
Cat.No: TP2206
Synonym: LEU 31, PRO34]-神经肽Y(猪)
Target: Neuropeptide Y Receptor
[Pro3]-GIP (Mouse) acetate
Cat.No: TP2020L
Synonym:
Target: Others
RO3244794
Cat.No: T69360
Synonym:
Target: Prostaglandin Receptor
Ro3280
Cat.No: T2634
Synonym: RO 3280,Ro5203280
Target: PLK
(Pro3) GIP, human
Cat.No: T76313
Synonym:
Target:
(Pro34)-Peptide YY (human)
Cat.No: T76441
Synonym:
Target:
RO320-2947/001
Cat.No: T34370
Synonym: RO-320-2947/001,RO 320-2947/001
Target:
[Pro3]-GIP (Rat)
Cat.No: TP2021
Synonym:
Target:
[Leu31,Pro34]-Neuropeptide Y(human,rat) TFA
Cat.No: T75912
Synonym:
Target:
[Leu31,Pro34]-Neuropeptide Y(human,rat)
Cat.No: TP1985
Synonym: [Leu31,Pro34]-Neuropeptide Y (human, rat)
Target:
[Pro3]-GIP (Mouse)
Cat.No: TP2020
Synonym:
Target:
TO-PRO3 iodide
Cat.No: T34903
Synonym: TOPRO3 iodide,TO-PRO3 iodide salt
Target:
RO314724
Cat.No: T71420
Synonym:
Target:
[D-Phe2,6, Pro3]-LH-RH
Cat.No: T83499
Synonym:
Target:
(Leu31,Pro34)-Peptide YY (human) (TFA)
Cat.No: T80087
Synonym:
Target: Neuropeptide Y Receptor
(Leu31,Pro34)-Peptide YY (human)
Cat.No: T76442
Synonym:
Target:
TargetMol Loading
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