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Cat. No. Product Name Target Signaling Pathways
T13675 Elacestrant dihydrochloride

RAD1901 dihydrochloride

Estrogen/progestogen Receptor Endocrinology/Hormones
Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) 是一种具有口服活性的的选择性雌激素受体 (ER) 降解剂 (SERD),能够作用于 ERα (IC50:48 nM) 和 ERβ (IC50:870 nM)。
T13674 Elacestrant

依拉司群,RAD1901

Estrogen Receptor/ERR; Estrogen/progestogen Receptor Endocrinology/Hormones
Elacestrant (RAD1901) 是一种具有口服活性的、选择性的雌激素受体 (ER) 降解剂 (SERD),能够作用于 ERα (IC50:48 nM)和 ERβ (IC50:870 nM)。
T11173L Elacestrant S enantiomer dihydrochloride

RAD1901 S enantiomer dihydrochloride,RAD-1901 S enantiomer dihydrochloride,RAD 1901 S enantiomer dihydrochloride

Others Others
Elacestrant (RAD1901) dihydrochloride is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively. Elacestrant S enantiomer dihydrochloride is an low activity enantiomer of elacestrant dihydrochloride.

化合物

Elacestrant dihydrochloride
Cat.No: T13675
Synonym: RAD1901 dihydrochloride
Target: Estrogen/progestogen Receptor
Elacestrant
Cat.No: T13674
Synonym: 依拉司群,RAD1901
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Elacestrant S enantiomer dihydrochloride
Cat.No: T11173L
Synonym: RAD1901 S enantiomer dihydrochloride,RAD-1901 S enantiomer dihydrochloride,RAD 1901 S enantiomer dihydrochloride
Target: Others
TargetMol Loading
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