Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1899 |
Pyridostatin
RR82,Pyridostatin Trifluoroacetate Salt |
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Pyridostatin (RR82) 是一种 G-四链体稳定剂,靶向原癌基因 Src,降低人乳腺癌细胞 SRC 蛋白水平和 SRC 依赖的细胞运动。它通过诱导复制和转录依赖的 DNA 损伤促进人类癌细胞生长停滞。 | |||
T4457 |
Pyridostatin Trihydrochloride
Pyridostatin Trihydrochloride(free base 1085412-37-8 ),RR-82 Trihydrochloride |
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Pyridostatin Trihydrochloride (RR-82 Trihydrochloride) 是一种 G-四链体稳定剂,Kd 为 490 nM。 | |||
T30745L |
Carboxy-pyridostatin 2HCl
Carboxy-pyridostatin 2HCl(1417638-60-8 Free base) |
DNA | DNA Damage/DNA Repair |
Carboxy-pyridostatin 2HCl 具有潜在的抗肿瘤活性,在 DNA G4s 上对 DNA 具有很高的亲和力。 | |||
T4470 |
Pyridostatin TFA
|
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Pyridostatin TFA 是一种 G-四链体稳定剂,靶向原癌基因 Src,降低人乳腺癌细胞 SRC 蛋白水平和 SRC 依赖的细胞运动。它通过诱导复制和转录依赖的 DNA 损伤促进人类癌细胞生长停滞。 | |||
T30745 |
Carboxy-pyridostatin
|
||
Carboxy-pyridostatin, as a fluorescent probe, can target G-quadruplex structures and trap cytoplasmic RNA G-quadruplex structures in cells. | |||
T72201 |
Pyridostatin hydrochloride
RR82 hydrochloride |
||
Pyridostatin (RR82) hydrochloride 是一种高选择性的 G-quadruplexDNA 稳定剂 (Kd=490 nM)。Pyridostatin hydrochloride 通过诱导复制和转录依赖的 DNA 损伤促进人类癌细胞生长停滞。Pyridostatin hydrochloride 靶向原癌基因 Src。Pyridostatin hydrochloride 降低人乳腺癌细胞 SRC 蛋白水平和 SRC 依赖的细胞运动。 | |||
T13595 |
Carboxy pyridostatin trifluoroacetate salt
|
Others | Others |
Carboxy pyridostatin trifluoroacetate salt exhibits higher molecular specificity for RNA over DNA G4s. |