Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T60636 |
Pitolisant
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Pitolisant 是一种有效的选择性的非咪唑类反相激动剂,作用于重组人组胺H3受体反相激动剂,Ki 值为 0.16 nM。 | |||
T7176 |
Pitolisant hydrochloride
1-[3-[3-(4-氯丙基)丙氧基]丙基]-哌啶盐酸盐,BF 2649,Ciproxidine |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Pitolisant hydrochloride (Ciproxidine) 是一种有效的、选择性的组胺 H3 受体反向激动剂,Ki 为0.16 nM。 | |||
T12491 |
Pitolisant oxalate
Tiprolisant oxalate |
Others | Others |
Pitolisant oxalate is a potent and selective inverse agonist of nonimidazole at the recombinant human histamine H3 receptor with Ki of 0.16 nM. |