Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12150 |
N-Methylbenzamide
|
PDE | Metabolism |
N-Methylbenzamide 是磷酸二酯酶 10A 抑制剂,具有抗癌作用。 | |||
T24656 |
PQ-10
A844337,PQ 10,A-844337,A 844337 |
PDE | Metabolism |
PQ-10 (A-844337) 是磷酸二酯酶 10A 抑制剂,其IC50=4.6 nM,ED50=13 mg/kg。它能够诱导大脑葡萄糖代谢模式,这可能是潜在的转化生物标志物。它对精神分裂症等精神疾病具有研究潜力。 | |||
T16499 |
Mardepodect
PF-2545920 |
PDE | Metabolism |
Mardepodect (PF-2545920) 是一种有效的、口服具有活性的、可透过血脑屏障的、选择性的 PDE10A 抑制剂,IC50=0.37 nM,比作用于其他 PDE 选择性高 1000 多倍。 | |||
T12119 |
MT-3014
|
Others | Others |
MT-3014 is a potent, highly selective and brain-penetrated inhibitor of phosphodiesterase 10A (PDE 10A)(human PDE 10A and bovine PDE 10A with IC50s of 0.062 nM and 0.09 nM , respectively). | |||
T32307 |
JNJ-42259152 F-18
|
||
JNJ-42259152 F-18 can be used as a Novel Phosphodiesterase 10A PET Tracer. | |||
T70761 |
ASP9436 Dihydrochloride
|
||
ASP9436 Dihydrochloride is a potent, selective and orally active phosphodiesterase 10A inhibitor. | |||
T28969 | THPP-4 | ||
THPP-4 inhibits phosphodiesterase 10A (PDE10A). | |||
T27684 |
JNJ-42259152
JNJ42259152,JNJ 42259152 |
||
JNJ-42259152 is a phosphodiesterase 10A PET tracer. | |||
T28968 |
THPP-2
|
||
HPP-2 is a novel phosphodiesterase 10A (PDE10A) inhibitor used to treat schizophrenia. | |||
T70822 |
Gemlapodect
RO554965 |
||
Gemlapodect (RO554965),一种针对磷酸二酯酶 10A (PDE10A) 的抑制剂,主要应用于精神分裂症的研究。 | |||
T23722 |
AMG-7980
AMG7980 |
||
AMG-7980 is a highly specific phosphodiesterase 10A ligand. It shows a good uptake in the striatum. | |||
T73462 | MK-8189 | ||
MK-8189 是一种口服有效的选择性PDE10A 抑制剂,Ki 值为 29 pM。MK-8189 可用于精神分裂症的研究。 |