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Cat. No. Product Name Target Signaling Pathways
T12150 N-Methylbenzamide

PDE Metabolism
N-Methylbenzamide 是磷酸二酯酶 10A 抑制剂,具有抗癌作用。
T24656 PQ-10

A844337,PQ 10,A-844337,A 844337

PDE Metabolism
PQ-10 (A-844337) 是磷酸二酯酶 10A 抑制剂,其IC50=4.6 nM,ED50=13 mg/kg。它能够诱导大脑葡萄糖代谢模式,这可能是潜在的转化生物标志物。它对精神分裂症等精神疾病具有研究潜力。
T16499 Mardepodect

PF-2545920

PDE Metabolism
Mardepodect (PF-2545920) 是一种有效的、口服具有活性的、可透过血脑屏障的、选择性的 PDE10A 抑制剂,IC50=0.37 nM,比作用于其他 PDE 选择性高 1000 多倍。
T12119 MT-3014

Others Others
MT-3014 is a potent, highly selective and brain-penetrated inhibitor of phosphodiesterase 10A (PDE 10A)(human PDE 10A and bovine PDE 10A with IC50s of 0.062 nM and 0.09 nM , respectively).
T32307 JNJ-42259152 F-18

JNJ-42259152 F-18 can be used as a Novel Phosphodiesterase 10A PET Tracer.
T70761 ASP9436 Dihydrochloride

ASP9436 Dihydrochloride is a potent, selective and orally active phosphodiesterase 10A inhibitor.
T28969 THPP-4

THPP-4 inhibits phosphodiesterase 10A (PDE10A).
T27684 JNJ-42259152

JNJ42259152,JNJ 42259152

JNJ-42259152 is a phosphodiesterase 10A PET tracer.
T28968 THPP-2

HPP-2 is a novel phosphodiesterase 10A (PDE10A) inhibitor used to treat schizophrenia.
T70822 Gemlapodect

RO554965

Gemlapodect (RO554965),一种针对磷酸二酯酶 10A (PDE10A) 的抑制剂,主要应用于精神分裂症的研究。
T23722 AMG-7980

AMG7980

AMG-7980 is a highly specific phosphodiesterase 10A ligand. It shows a good uptake in the striatum.
T73462 MK-8189

MK-8189 是一种口服有效的选择性PDE10A 抑制剂,Ki 值为 29 pM。MK-8189 可用于精神分裂症的研究。

化合物

N-Methylbenzamide
Cat.No: T12150
Synonym:
Target: PDE
PQ-10
Cat.No: T24656
Synonym: A844337,PQ 10,A-844337,A 844337
Target: PDE
Mardepodect
Cat.No: T16499
Synonym: PF-2545920
Target: PDE
MT-3014
Cat.No: T12119
Synonym:
Target: Others
JNJ-42259152 F-18
Cat.No: T32307
Synonym:
Target:
ASP9436 Dihydrochloride
Cat.No: T70761
Synonym:
Target:
THPP-4
Cat.No: T28969
Synonym:
Target:
JNJ-42259152
Cat.No: T27684
Synonym: JNJ42259152,JNJ 42259152
Target:
THPP-2
Cat.No: T28968
Synonym:
Target:
Gemlapodect
Cat.No: T70822
Synonym: RO554965
Target:
AMG-7980
Cat.No: T23722
Synonym: AMG7980
Target:
MK-8189
Cat.No: T73462
Synonym:
Target:
TargetMol Loading
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