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Search Results for " ppar-alpha "
Targets Recommended: PPAR

9

抑制剂 & 化合物

2

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T16022 Arhalofenate

JNJ 39659100,芳卤芬酯,4-氯-ALPHA-[3-(三氟甲基)苯氧基]苯乙酸 2-(乙酰基氨基)乙酯,MBX 102

PPAR DNA Damage/DNA Repair; Metabolism
Arhalofenate (JNJ 39659100) 是一种选择性的(PPAR)-γ部分激动剂,用于研究 2 型糖尿病。
T27706 K-111

BM170744,BM 170744,BM-170744,K111

K-111 is a PPAR alpha agonist. K-111 improves insulin resistance, reducing bodyweight, and ameliorating atherogenic dyslipidemia.
T15575 Indeglitazar

PPM 204

PPAR DNA Damage/DNA Repair; Metabolism
Indeglitazar (PPM 204) 是 PPAR 的泛激动剂,包括亚型 alpha (α)、delta (δ) 和 gamma (γ)。
T5532 BMS-687453

PPAR DNA Damage/DNA Repair; Metabolism
BMS-687453 是一种选择性 PPARα激动剂,对人 PPARα的 EC50和 IC50分别为 10 nM 和 260 nM。它较弱地抑制 PPARγ 的活性,EC50和 IC50值分别为 4100 nM 和大于 15000 nM。
T10900 CUDA

PPAR; Epoxide Hydrolase DNA Damage/DNA Repair; Metabolism
CUDA 是一种可溶性环氧水解酶抑制剂,对小鼠 sEH 和人 sEH 作用的 IC50分别为 11.1 和 112 nM。它能选择性地上调过氧化物酶体增殖激活受体 PPARα的活性,有用于心血管疾病的研究潜力。
T27508 GW409544

GW 409544,GW-409544

GW409544 is an agonist of PPAR-alpha and PPAR-gamma.
T27208 DRF 2519

DRF2519,DRF-2519

DRF 2519 is an activator of PPAR-alpha and PPAR-gamma.
T29028 TZD18

TZD-18,TZD 18

TZD18, a novel PPAR alpha/gamma dual agonist, inhibits cell growth and induces apoptosis in human glioblastoma T98G cells.
T69191 Pemaglitazar

Pemaglitazar is a dual peroxisome proliferator-activated receptor (PPAR) alpha and gamma agonist, with hypoglycemic activity.

化合物

Arhalofenate
Cat.No: T16022
Synonym: JNJ 39659100,芳卤芬酯,4-氯-ALPHA-[3-(三氟甲基)苯氧基]苯乙酸 2-(乙酰基氨基)乙酯,MBX 102
Target: PPAR
K-111
Cat.No: T27706
Synonym: BM170744,BM 170744,BM-170744,K111
Target:
Indeglitazar
Cat.No: T15575
Synonym: PPM 204
Target: PPAR
BMS-687453
Cat.No: T5532
Synonym:
Target: PPAR
CUDA
Cat.No: T10900
Synonym:
Target: PPAR, Epoxide Hydrolase
GW409544
Cat.No: T27508
Synonym: GW 409544,GW-409544
Target:
DRF 2519
Cat.No: T27208
Synonym: DRF2519,DRF-2519
Target:
TZD18
Cat.No: T29028
Synonym: TZD-18,TZD 18
Target:
Pemaglitazar
Cat.No: T69191
Synonym:
Target:
Cat. No. Product Name Species Expression System
TMPY-06837 PPAR alpha/PPARA Protein, Mouse, Recombinant (His)

PPARα,PPAR-alpha,peroxisome proli...

Mouse E. coli
PPAR alpha/PPARA Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 31.49 kDa and the accession number is P23204.
TMPY-06830 PPAR alpha/PPARA Protein, Human, Recombinant (His)

NR1C1,PPARα,peroxisome proliferator-activated recep...

Human E. coli
PPAR alpha/PPARA Protein, Human, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 31.36 kDa and the accession number is Q07869.

重组蛋白

PPAR alpha/PPARA Protein, Mouse, Recombinant (His)
Cat.No: TMPY-06837
Species: Mouse
Expression System: E. coli
PPAR alpha/PPARA Protein, Human, Recombinant (His)
Cat.No: TMPY-06830
Species: Human
Expression System: E. coli
TargetMol Loading
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