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2
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T16022 |
Arhalofenate
JNJ 39659100,芳卤芬酯,4-氯-ALPHA-[3-(三氟甲基)苯氧基]苯乙酸 2-(乙酰基氨基)乙酯,MBX 102 |
PPAR | DNA Damage/DNA Repair; Metabolism |
Arhalofenate (JNJ 39659100) 是一种选择性的(PPAR)-γ部分激动剂,用于研究 2 型糖尿病。 | |||
T27706 |
K-111
BM170744,BM 170744,BM-170744,K111 |
||
K-111 is a PPAR alpha agonist. K-111 improves insulin resistance, reducing bodyweight, and ameliorating atherogenic dyslipidemia. | |||
T15575 |
Indeglitazar
PPM 204 |
PPAR | DNA Damage/DNA Repair; Metabolism |
Indeglitazar (PPM 204) 是 PPAR 的泛激动剂,包括亚型 alpha (α)、delta (δ) 和 gamma (γ)。 | |||
T5532 |
BMS-687453
|
PPAR | DNA Damage/DNA Repair; Metabolism |
BMS-687453 是一种选择性 PPARα激动剂,对人 PPARα的 EC50和 IC50分别为 10 nM 和 260 nM。它较弱地抑制 PPARγ 的活性,EC50和 IC50值分别为 4100 nM 和大于 15000 nM。 | |||
T10900 |
CUDA
|
PPAR; Epoxide Hydrolase | DNA Damage/DNA Repair; Metabolism |
CUDA 是一种可溶性环氧水解酶抑制剂,对小鼠 sEH 和人 sEH 作用的 IC50分别为 11.1 和 112 nM。它能选择性地上调过氧化物酶体增殖激活受体 PPARα的活性,有用于心血管疾病的研究潜力。 | |||
T27508 |
GW409544
GW 409544,GW-409544 |
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GW409544 is an agonist of PPAR-alpha and PPAR-gamma. | |||
T27208 |
DRF 2519
DRF2519,DRF-2519 |
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DRF 2519 is an activator of PPAR-alpha and PPAR-gamma. | |||
T29028 |
TZD18
TZD-18,TZD 18 |
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TZD18, a novel PPAR alpha/gamma dual agonist, inhibits cell growth and induces apoptosis in human glioblastoma T98G cells. | |||
T69191 |
Pemaglitazar
|
||
Pemaglitazar is a dual peroxisome proliferator-activated receptor (PPAR) alpha and gamma agonist, with hypoglycemic activity. |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-06837 |
PPAR alpha/PPARA Protein, Mouse, Recombinant (His)
PPARα,PPAR-alpha,peroxisome proli... |
Mouse | E. coli |
PPAR alpha/PPARA Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 31.49 kDa and the accession number is P23204. | |||
TMPY-06830 |
PPAR alpha/PPARA Protein, Human, Recombinant (His)
NR1C1,PPARα,peroxisome proliferator-activated recep... |
Human | E. coli |
PPAR alpha/PPARA Protein, Human, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 31.36 kDa and the accession number is Q07869. |