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Cat. No. Product Name Target Signaling Pathways
T79241 PHD2-IN-1

HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism
PHD2-IN-1 为一种口服活性强效 HIF-脯氨酰羟化酶2 (PHD2) 抑制剂,具有 22.53 nM 的 IC50 值,适用于贫血病研究。
T62298 PHD2/HDACs-IN-1

PHD2/HDACs-IN-1 是一种有效的 PHD2/HDACs 混合抑制剂,能够作用于 PHD2 (IC50: 1.15 μM)、HDAC1 (IC50: 19.75 μM)、HDAC2 (IC50: 26.60 μM)、HDAC16 (IC50: 15.98 μM)。PHD2/HDACs-IN-1 是一种低毒性肾保护剂,能够用于顺铂诱导的急性肾损伤 (AKI) 的研究。
T1823 IOX2

IOX 2,JICL38

HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism
IOX2 (IOX 2) 是特异性的脯氨酰羟化酶-2 抑制剂,IC50=22 nM。
T79797 PHD-IN-1

HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism
PHD-IN-1(compound 80)作为PHD2的抑制剂,显示出 IC50 ≤5 nM 的高效活性。在Caco2-HIFla-HiBiT-clone-1和Hep3B细胞系中进行的EPO Elisa实验中,其EC50值均为2.5 μM。
T61458 HIF-PHD-IN-2

HIF-PHD-IN-2 (compound 25) is a highly effective PHD inhibitor, displaying IC50 values below 100 nM for PHD1, PHD2, and PHD3 [1].
T39040 HIF-PHD-IN-1

HIF-PHD-IN-1 is a pharmacological compound that acts as an orally active inhibitor of the hypoxia-inducible factor prolyl hydroxylase domain (HIF-PHD), displaying an IC50 of 54 nM for hHIF-PHD2. Its potential as a therapeutic agent for renal anemia is highly promising.
T68511 KRH102140

KRH102140 is a potent activator of PHD2. KRH102140, which has a structure similar to KRH102053. KRH102140 more efficiently suppressed HIF-1α than KRH102053 in human osteosarcoma cells under hypoxia. Furthermore, KRH102140 decreased the mRNA levels of HIF-regulated downstream target genes associated with angiogenesis and energy metabolism such as vascular endothelial growth factor, adrenomedullin, Glut1, aldolase A, enolase 1 and monocarboxylate transporter 4. KRH102140 also inhibited tube format...

化合物

PHD2-IN-1
Cat.No: T79241
Synonym:
Target: HIF/HIF Prolyl-Hydroxylase
PHD2/HDACs-IN-1
Cat.No: T62298
Synonym:
Target:
IOX2
Cat.No: T1823
Synonym: IOX 2,JICL38
Target: HIF/HIF Prolyl-Hydroxylase
PHD-IN-1
Cat.No: T79797
Synonym:
Target: HIF/HIF Prolyl-Hydroxylase
HIF-PHD-IN-2
Cat.No: T61458
Synonym:
Target:
HIF-PHD-IN-1
Cat.No: T39040
Synonym:
Target:
KRH102140
Cat.No: T68511
Synonym:
Target:
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