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Cat. No. Product Name Target Signaling Pathways
T4171 PEAQX

NVP-AAM077

NMDAR; iGluR Membrane transporter/Ion channel; Neuroscience
PEAQX (NVP-AAM077) 是 NR2A 高效选择性 NMDA 受体拮抗剂,IC50值为270nM。
T16451 PEAQX tetrasodium hydrate

NVP-AAM077 tetrasodium hydrate,PEAQX tetrasodium hydrate (459836-30-7 free base),PEAQX tetrasodium hydrate

Apoptosis; NMDAR; iGluR Apoptosis; Membrane transporter/Ion channel; Neuroscience
PEAQX tetrasodium hydrate (PEAQX tetrasodium hydrate (459836-30-7 free base)) 是一种可口服的NMDA 拮抗剂,具有有效性和选择性。PEAQX tetrasodium hydrate (459836-30-7 free base) 对 hNMDAR 1A/2A 的 IC50 值分别为 270 nM 对hNMDAR 1A/2B 的 IC50 值为29600 nM。
T69906 PEAQX sodium

PEAQX, also known as NVP-AAM077; is a competitive antagonist at the NMDA receptor. Although originally described as 100-fold selective for GluN1/GluN2A receptors vs. GluN1/GluN2B receptors, more detailed studies of the Ki of PEAQX revealed it only shows a 5 fold difference in affinity for GluN1/GluN2A vs. GluN1/GluN2B receptors. It is also a potent anticonvulsant in animal tests.
T69905 Iferanserin HCl

Iferanserin HCl is a selective serotonin receptor antagonist.

化合物

PEAQX
Cat.No: T4171
Synonym: NVP-AAM077
Target: NMDAR, iGluR
PEAQX tetrasodium hydrate
Cat.No: T16451
Synonym: NVP-AAM077 tetrasodium hydrate,PEAQX tetrasodium hydrate (459836-30-7 free base),PEAQX tetrasodium hydrate
Target: Apoptosis, NMDAR, iGluR
PEAQX sodium
Cat.No: T69906
Synonym:
Target:
Iferanserin HCl
Cat.No: T69905
Synonym:
Target:
TargetMol Loading
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