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Search Results for " pde5a "

6

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T27122 Dasantafil

SCH446132,SCH-446132,SCH 446132

PDE Metabolism
Dasantafil (SCH446132) 是一种小分子磷酸二酯酶-5A(PDE5A)抑制剂,可用于治疗泌尿生殖系统疾病和研究勃起功能障碍。
T15381 Gisadenafil

UK-369003,吉沙那非

PDE Metabolism
Gisadenafil (UK-369003) 是一种特异性磷酸二酯酶 5 (PDE5) 抑制剂,IC50 为 3.6 nM,可防止 cGMP 降解。
T27720 KD-027

KD 027,SLx-2101,SLx2101,KD027,SLx 2101

KD-027, a PDE5A inhibitor, is used potentially for the treatment of hypertension.
T29048 UK 357903

UK357903,UK-357903

UK 357903, a phosphodiesterase 5A (PDE5A) inhibitor, is used potentially for the treatment of erectile dysfunction.
T28296 Parogrelil hydrochloride

INDI-702,NM-702,NT-702,NM702,INDI702

Parogrelil is a phosphodiesterase (PDE3/PDE5A) inhibitor potentially for the treatment of intermittent. Parogrelil suppress the asthmatic response in guinea pigs, with both bronchodilating and anti-inflammatory effects. Parogrelil improves reduced walking
T11400 Gisadenafil besylate

UK 369003-26

Others Others
Gisadenafil besylate (UK 369003-26) is a specific, orally active phosphodiesterase 5 (PDE5) inhibitor ,prevents degradation of cyclic guanosine monophosphate (cGMP), with an IC50 of 3.6 nM .

化合物

Dasantafil
Cat.No: T27122
Synonym: SCH446132,SCH-446132,SCH 446132
Target: PDE
Gisadenafil
Cat.No: T15381
Synonym: UK-369003,吉沙那非
Target: PDE
KD-027
Cat.No: T27720
Synonym: KD 027,SLx-2101,SLx2101,KD027,SLx 2101
Target:
UK 357903
Cat.No: T29048
Synonym: UK357903,UK-357903
Target:
Parogrelil hydrochloride
Cat.No: T28296
Synonym: INDI-702,NM-702,NT-702,NM702,INDI702
Target:
Gisadenafil besylate
Cat.No: T11400
Synonym: UK 369003-26
Target: Others
Cat. No. Product Name Target Signaling Pathways
TN2159 Robustine

大叶桉亭,8-羟基白鲜碱,4-甲氧基呋喃并[2,3-B]喹啉-8-醇

PDE Metabolism
Robustine 是一种从 Dictamnus albus 获得的呋喃喹啉生物碱,在体外对人磷酸二酯酶 5 (hPDE5A) 具有抑制作用。
T38108 Fulvic Acid

Antioxidant; PDE Metabolism; oxidation-reduction
Fulvic Acid 是一种来自土壤、沉积物或水生环境中微生物产生的腐殖质的天然产物,是一种首次青霉菌中分离出的酚酸和真菌代谢产物。Fulvic Acid 抑制淀粉样蛋白b (17-42) (AB17-42)二聚化,破坏预先形成的AB17-42三聚体,并结合到磷酸二酯酶5A (PDE5A)的催化位点,可以调节机体免疫系统,影响细胞的氧化状态,改善胃肠功能。Fulvic Acid 可作为氧化剂或还原剂, 具有研究糖尿病等慢性炎症性疾病的潜力。

天然产物

Robustine
Cat.No: TN2159
Synonym: 大叶桉亭,8-羟基白鲜碱,4-甲氧基呋喃并[2,3-B]喹啉-8-醇
Target: PDE
Fulvic Acid
Cat.No: T38108
Synonym:
Target: Antioxidant, PDE
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