Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3063 |
PD173955
PD-173955,PD 173955 |
Apoptosis; Bcr-Abl; Src | Angiogenesis; Apoptosis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors |
PD173955是一种Src 激酶家族选择性抑制剂,对Src、Yes 和Abl 激酶IC50值约为22nM, 对 FGFRα 的效力较低,对InsR 和PKC 无活性。 | |||
T71912 |
PD 173955-Analog1
|
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PD 173955-Analog1 is a potent c-Src inhibitor known to have activity against a variety of cancers including colon, lung, head and neck carcinoma. |