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Cat. No. Product Name Target Signaling Pathways
T16440 Ibrutinib Racemate

PCI-32765 (Racemate)

Others Others
Ibrutinib is a selective, irreversible Btk inhibitor (IC50: 0.5 nM). Ibrutinib Racemate is the racemate of Ibrutinib.
T13814 Pemafibrate (racemate)

K13675 (racemate)

Others Others
Pemafibrate racemate is the racemate of pemafibrate
T13450L GNE-140 racemate

GNE-140 (racemate)

Others Others
GNE-140 is a potent inhibitor of lactate dehydrogenase A (LDHA). GNE-140 is a racemate mixture of (R)-GNE-140 and (S)-GNE-140.
T1835 Ibrutinib

伊布替尼,依鲁替尼,PCI-32765

Tyrosine Kinases; Src; BTK; Ligands for Target Protein for PROTAC Angiogenesis; PROTAC; Tyrosine Kinase/Adaptors
Ibrutinib (PCI-32765) 是一种不可逆的、选择性的 Btk 抑制剂,IC50=0.5 nM,它是一种 Btk 配体,用于合成一系列 PROTAC 分子,如 P13I。P13I 作用于人 Burkitt’s 淋巴瘤 RAMOS 细胞,浓度为 10 和 100 nM 时,分别降解 73% 和 89% Btk。

化合物

Ibrutinib Racemate
Cat.No: T16440
Synonym: PCI-32765 (Racemate)
Target: Others
Pemafibrate (racemate)
Cat.No: T13814
Synonym: K13675 (racemate)
Target: Others
GNE-140 racemate
Cat.No: T13450L
Synonym: GNE-140 (racemate)
Target: Others
Ibrutinib
Cat.No: T1835
Synonym: 伊布替尼,依鲁替尼,PCI-32765
Target: Tyrosine Kinases, Src, BTK, Ligands for Target Protein for PROTAC
TargetMol Loading
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