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Cat. No. Product Name Target Signaling Pathways
T6916 OICR-9429

OICR 9429

Histone Methyltransferase; JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
OICR-9429 是一个新颖的相互作用的小分子Wdr5-MLL 拮抗剂,IC50是 5 uM,在体外抑制急性髓性白血病细胞。
T39978 Dimethyl-F-OICR-9429-COOH

Dimethyl-F-OICR-9429-COOH, a ligand for WD40 repeat domain protein 5 (WDR5). This compound is utilized as a key component in the synthesis of PROTACs.
T39977 OICR-9429-N-C2-NH2

OICR-9429-N-C2-NH2

OICR-9429-N-C2-NH2, a ligand for WDR5, intermediate 2, serves as a crucial compound in the synthesis of PROTACs.
T77495 WDR5-IN-6

JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
WDR5-IN-6 是一种 WDR5 抑制剂,靶向 WBM 位点。WDR5-IN-6 与靶向 WIN 位点的 WDR5 抑制剂 OICR-9429 具有高度协同作用。WDR5-IN-6 具有较强的抗肿瘤活性,可抑制神经母细胞瘤细胞系的细胞增殖。WDR5-IN-6 可用于神经母细胞瘤的研究。
T12290 OICR-0547

Others Others
OICR-0547 is a closely related derivative of OICR-9429. OICR-9429 is a novel small-molecule Wdr5-MLL interaction antagonist.

化合物

OICR-9429
Cat.No: T6916
Synonym: OICR 9429
Target: Histone Methyltransferase, JAK
Dimethyl-F-OICR-9429-COOH
Cat.No: T39978
Synonym:
Target:
OICR-9429-N-C2-NH2
Cat.No: T39977
Synonym: OICR-9429-N-C2-NH2
Target:
WDR5-IN-6
Cat.No: T77495
Synonym:
Target: JAK
OICR-0547
Cat.No: T12290
Synonym:
Target: Others
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