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Cat. No. Product Name Target Signaling Pathways
T10358 Netarsudil Dihydrochloride

AR-13324 Dihydrochloride

ROCK Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
Netarsudil Dihydrochloride (AR-13324 Dihydrochloride) 是 Rho 相关蛋白激酶 (ROCK) 和去甲肾上腺素转运蛋白 (NET) 的抑制剂,可有效降低眼压 (IOP)。
T10358L2 Netarsudil mesylate

AR-13324 (mesylate)

Others Others
Netarsudil mesylate is an inhibitor of Rho-associated protein kinase (ROCK) and norepinephrine transporter (NET) with effective in intraocular pressure (IOP) reduction.
T71119 Netarsudil free base

Netarsudil, also known as AR-11324, is a Rho-associated protein kinase inhibitor. Netarsudil is potential useful for treating glaucoma and​/or reducing intraocular pressure. Netarsudil Increases Outflow Facility in Human Eyes Through Multiple Mechanisms. Netarsudil inhibited kinases ROCK1 and ROCK2 with a Ki of 1 nM each, disrupted actin stress fibers and focal adhesions in TM cells with IC50s of 79 and 16 nM, respectively, and blocked the profibrotic effects of TGF-β2 in HTM cells. Netarsudi...
T71973 Gilteritinib hemifumarate

ASP2215 hemifumarate

FLT; TAM Receptor Angiogenesis; Tyrosine Kinase/Adaptors
Gilteritinib hemifumarate (ASP2215 hemifumarate) 是一种高效的 ATP 竞争性 FLT3(IC50 : 0.29 nM) 和 AXL(IC50: 0.73 nM) 双重抑制剂,可用于治疗复发或难治性 FLT3 突变的 AML。
T71118 NEP-28

NEP-28 is an AR agonist. NEP28 is a new SARM exhibiting high selectivity for androgen receptor. NEP28 showed tissue-selective effect equivalent to or higher than existing SARMs. In addition, the administration of NEP28 increased the activity of neprilysin, a known Aβ-degrading enzyme.
T71120 AR-13503

AR-13503, is an metabolite of Netarsudil (AR-11324), is a Rho-associated protein kinase inhibitor. Netarsudil is potential useful for treating glaucoma and​/or reducing intraocular pressure.

化合物

Netarsudil Dihydrochloride
Cat.No: T10358
Synonym: AR-13324 Dihydrochloride
Target: ROCK
Netarsudil mesylate
Cat.No: T10358L2
Synonym: AR-13324 (mesylate)
Target: Others
Netarsudil free base
Cat.No: T71119
Synonym:
Target:
Gilteritinib hemifumarate
Cat.No: T71973
Synonym: ASP2215 hemifumarate
Target: FLT, TAM Receptor
NEP-28
Cat.No: T71118
Synonym:
Target:
AR-13503
Cat.No: T71120
Synonym:
Target:
TargetMol Loading
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