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Cat. No. Product Name Target Signaling Pathways
T70198 Atrasentan sodium

Atrasentan, also known as ABT-627, is a orally available ETA receptor antagonist with potential antineoplastic activity. As a selective antagonist of the endothelin-A (ETA) receptor, atrasentan binds selectively to the ETA receptor, which may result in inhibition of endothelin-induced angiogenesis and tumor cell proliferation.
T6481 Droxinostat

NS 41080,4-(4-氯-2-甲基苯氧基)-N-羟基丁酰胺

Apoptosis; HDAC Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair
Droxinostat (NS 41080) 是HDAC3、HDAC6和HDAC8抑制剂,IC50分别为16.9、2.47和1.46 μM。
T38779 NS-102

NS-102 is a powerful and selective antagonist of the kainate receptor (GluK2), as well as a potent antagonist of the GluR6/7 receptor.
T36905 Nanangenine F

Nanangenine F is a drimane sesquiterpene fungal metabolite that has been found inA. nanangensis.1It is active againstB. subtilis(IC50= 78 μg/ml) and cytotoxic to NS-1, DU145, and MCF-7 cancer and NFF non-cancerous cells (IC50s = 49, 95, 49, and 84 μg/ml, respectively). 1.Lacey, H.J., Gilchrist, C.L.M., Crombie, A., et al.Nanangenines: Drimane sesquiterpenoids as the dominant metabolite cohort of a novel Australian fungus, Aspergillus nanangensisBeilstein J. Org. Chem.152631-2643(2019)

化合物

Atrasentan sodium
Cat.No: T70198
Synonym:
Target:
Droxinostat
Cat.No: T6481
Synonym: NS 41080,4-(4-氯-2-甲基苯氧基)-N-羟基丁酰胺
Target: Apoptosis, HDAC
NS-102
Cat.No: T38779
Synonym:
Target:
Nanangenine F
Cat.No: T36905
Synonym:
Target:
TargetMol Loading
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