Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11641 |
N-Desmethyl imatinib
Imatinib metabolite N-Desmethyl imatinib,Norimatinib,N-去甲基伊马替尼 |
Bcr-Abl; PDGFR; c-Kit; Drug Metabolite | Angiogenesis; Cytoskeletal Signaling; Metabolism; Tyrosine Kinase/Adaptors |
N-Desmethyl imatinib (Imatinib metabolite N-Desmethyl imatinib) 是 Imatinib 的代谢物。Imatinib 是一个靶向 c-Kit、v-Abl 和 PDGFR 的多靶点抑制剂。 | |||
T40504 |
N-Desmethyl imatinib mesylate
ImatinibmetaboliteN-Desmethylimatinibmesylate,N-Desmethyl imatinib mesylate,Norimatinib mesylate |
||
Norimatinib mesylate, also known as N-Desmethyl imatinib mesylate, is a metabolite derived from Imatinib, which acts as a potent multi-target inhibitor of v-Abl, c-Kit, and PDGFR. | |||
T19451 |
N-Desmethyl imatinib-d8
Norimatinib D8,Imatinib metabolite N-Desmethyl imatinib D8,N-Desmethyl imatinib D8 |
Others | Others |
N-Desmethyl imatinib D8 is a deuterium labeled Imatinib metabolite N-Desmethyl Imatinib. |