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Search Results for " nci-n87 "

4

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T6442 CH5138303

HSP Cytoskeletal Signaling; Metabolism
CH5138303 是一种可口服的 Hsp90 抑制剂,Kd 为 0.48 nM。
T34602 Selatinib

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Selatinib 是一种具有口服活性和有效性的 EGFR 和 ErbB2 双重抑制剂,具有抗癌活性,抑制 NCI-N87 肿瘤细胞生长。
T82802 BX-2819

HSP Cytoskeletal Signaling; Metabolism
BX-2819为一种Hsp90抑制剂,具有41 nM 的IC50值,能有效抑制癌细胞增殖,并在裸鼠模型中显著抑制NCI-N87和HT-29肿瘤生长。
T36684 Ipivivint

Ipivivint, a first-in-class, orally active and potent CDC-like kinase (CLK) inhibitor, inhibits CLK1 (IC50=1.4 μM), CLK2 (IC50=0.002 μM) and CLK3 (IC50=0.022 μM). Ipivivint reduces Wnt pathway signaling gene expression through inhibiting CLK activity and serine and arginine rich splicing factor (SRSF) phosphorylation and disrupting spliceosome activity. Ipivivint can be used for the research of cancer[1]. Ipivivint (SW480 cells; 0.01~10 μM; 1 hour) potently inhibits SRSF5/6 phosphorylation[1].Ip...

化合物

CH5138303
Cat.No: T6442
Synonym:
Target: HSP
Selatinib
Cat.No: T34602
Synonym:
Target: EGFR
BX-2819
Cat.No: T82802
Synonym:
Target: HSP
Ipivivint
Cat.No: T36684
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN3495 Benzyl ferulate

TNF; Antifection Apoptosis; Microbiology/Virology
Benzyl ferulate has antimicrobial activity. It also shows good anti-proliferative against three gastro-intestinal cancer cell lines(HCT-116 colon carcinoma, KYSE-30 oesophageal squamous cancer, and NCI-N87 gastric carcinoma).

天然产物

Benzyl ferulate
Cat.No: TN3495
Synonym:
Target: TNF, Antifection
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