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Cat. No.	Product Name	Target	Signaling Pathways
T81792	Mip-IN-1
	Mip-IN-1（S,S-28i）是一款新型雷帕霉素衍生的Mip抑制剂，对Neisseria meningitidis和Neisseria gonorrhoeae的Mip蛋白具有高效的抗酶作用，能显著增强巨噬细胞杀灭细菌的能力。
T7499	TAK-779 Takeda 779	HIV Protease; CXCR; CCR	Autophagy; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
	TAK-779 (Takeda 779) 是一种非肽类CCR5和CXCR3 拮抗剂，对CCR5的Ki 值为 1.1 nM，并选择性抑制R5 HIV-1。
T80977	TLR4 agonist-1 TEA
	TLR4agonist-1 (TEA) (compound 17a)为Toll-like Receptor 4 (TLR4)的高效激动剂，在RAW 264.7及MM6细胞中能有效促进MIP-1β的生成。
T80978	TLR4 agonist-1
	TLR4agonist-1 (compound 17a)是一种针对Toll-like Receptor 4 (TLR4)的高效激动剂，能有效激发RAW 264.7与MM6细胞产生MIP-1β。
T80090	Lugdunin	Antibiotic	Microbiology/Virology
	Lugdunin是一种具有抗菌活性的肽类抗生素。该化合物能够通过破坏细菌细胞膜的电位来抑制革兰氏阳性菌的生长，特别是对金黄色葡萄球菌（Staphylococcus aureus）表现出高效能，有效降低其在皮肤和鼻腔的定植能力。此外，Lugdunin还能在人类角质形成细胞和小鼠皮肤中促进LL-37和CXCL8/MIP-2的表达。
T81708	Nagrestipen
	Nagrestipen 是一种人巨噬细胞炎症蛋白-1α 变体，也称为 ECI 301，主要用于癌症、肿瘤、转移、放射肿瘤学以及肿瘤转移研究试验，具有显著的抗肿瘤活性。
T16973	TAK-220	HIV Protease	Microbiology/Virology; Proteases/Proteasome
	TAK-220 is a selective and orally bioavailable CCR5 antagonist (IC50s: 3.5 nM and 1.4 nM for inhibition on the binding of RANTES and MIP-1α to CCR5, respectively).
T37861	Talabostat
	Talabostat (PT100, Val-boroPro) is a potent, nonselective and orally available dipeptidyl peptidase IV (DPP-IV) inhibitor with a Ki of 0.18 nM. Talabostat is a nonselective DPP-IV inhibitor, inhibiting DPP8/9, FAP, DPP2 and some other DASH family enzymes essentially as potently as it inhibits DPP-IV[1]. Talabostat stimulates the immune system by triggering a proinflammatory form of cell death in monocytes and macrophages known as pyroptosis. The inhibition of two serine proteases, DPP8 and DPP9,...
T35451	β-Defensin-2 (human) (trifluoroacetate salt)
	β-Defensin-2 is a peptide with antimicrobial properties that protects the skin and mucosal membranes of the respiratory, genitourinary, and gastrointestinal tracts.1It inhibits the growth of periodontopathogenic and cariogenic bacteria, includingP. gingivalisandS. salivarius.2β-Defensin-2 (30 μg/ml) stimulates gene expression and production of IL-6, IL-10, CXCL10, CCL2, MIP-3α, and RANTES by keratinocytes.3It also stimulates calcium mobilization, migration, and proliferation of keratinocytes whe...