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Cat. No. Product Name Target Signaling Pathways
T20028 Janumet

Efficib,Janumet XR,Metformin / sitagliptin,Metformin hydrochloride mixture with sitagliptin phosphate

Metformin hydrochloride mixture with sitagliptin phosphate is an AMP-activated protein kinase stimulant. It is also a CD26 antigen inhibitor, Gluconeogenesis inhibitor, and Glucose modulator.
T0242 Sitagliptin

西他列汀,MK0431,西格列汀

Proteasome; DPP-4; Autophagy Autophagy; Proteases/Proteasome; Ubiquitination
Sitagliptin (MK0431) 是一种有效的 DPP4抑制剂,在 Caco-2 细胞中,IC50值为 19 nM。它是一种新型口服降糖药,可单独使用或与二甲双胍或噻唑烷二酮联合用于治疗 2 型糖尿病。

化合物

Janumet
Cat.No: T20028
Synonym: Efficib,Janumet XR,Metformin / sitagliptin,Metformin hydrochloride mixture with sitagliptin phosphate
Target:
Sitagliptin
Cat.No: T0242
Synonym: 西他列汀,MK0431,西格列汀
Target: Proteasome, DPP-4, Autophagy
TargetMol Loading
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