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Cat. No. Product Name Target Signaling Pathways
T22361 Mepivacaine

Carbocaine

Sodium Channel Membrane transporter/Ion channel
Mepivacaine (Carbocaine) 是一种可用于局部麻醉的酰胺类化合物,可使人或动物短暂的失去自知觉。Mepivacaine 通过与神经细胞膜上特定的电压门控钠离子通道结合,抑制钠离子内流和膜去极化来发挥作用。Mepivacaine 适用于神经阻滞和硬膜外麻醉。
T0946 Mepivacaine hydrochloride

Mepivacaine HCl,盐酸甲哌卡因

Sodium Channel Membrane transporter/Ion channel
Mepivacaine hydrochloride (Mepivacaine HCl) 是具有局部麻醉特性的酰胺衍生物。Mepivacaine hydrochloride 与神经元细胞膜上特定的电压门控钠离子通道结合,抑制钠离子内流和膜去极化。
T31400 Dexivacaine

BRN-0211230,Dexivacaina,BRN0211230,L(+)-Mepivacaine,BRN 0211230

Dexivacaine is an type of anesthetic.
T2131 Articaine hydrochloride

Ultracaine,盐酸阿替卡因,阿替卡因,Articaine HCl,Hoe-045

Sodium Channel Membrane transporter/Ion channel
Articaine hydrochloride (Hoe-045) 一种牙科局部麻醉剂。
T70538 PD-85639

PD-85639 is a voltage-gated sodium (Na+) channel blocker (75% in 10 min & >95% in 25 min blockage of Na+ current by 25 μM PD85,639; whole-cell patch clamp using primary rat brain neurons) that is shown to target rat brain Nav1.2 with simultaneous high- and low-affinity modes of binding (EC50 = 56 nM/40% & 20 μM/60% at pH 9.0, 5 nM/28% & 3 μM/72% at pH 7.4, against 2 nM [3H]-PD85,639 for binding rat brain synaptosomes; EC50 = 17 nM/39% & 10 μM/61% using at pH 9.0 using rat brain synaptosome membr...

化合物

Mepivacaine
Cat.No: T22361
Synonym: Carbocaine
Target: Sodium Channel
Mepivacaine hydrochloride
Cat.No: T0946
Synonym: Mepivacaine HCl,盐酸甲哌卡因
Target: Sodium Channel
Dexivacaine
Cat.No: T31400
Synonym: BRN-0211230,Dexivacaina,BRN0211230,L(+)-Mepivacaine,BRN 0211230
Target:
Articaine hydrochloride
Cat.No: T2131
Synonym: Ultracaine,盐酸阿替卡因,阿替卡因,Articaine HCl,Hoe-045
Target: Sodium Channel
PD-85639
Cat.No: T70538
Synonym:
Target:
TargetMol Loading
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