Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T16040 |
Mepazine
甲哌啶嗪,Pecazine |
Apoptosis; MALT | Apoptosis; Immunology/Inflammation |
Mepazine (Pecazine) 是一种有效的特异性 MALT1 抑制剂。 Mepazine 抑制 GSTMALT1 全长和 GSTMALT1 325-760,IC50 为 0.83 μM 和 0.42 μM。 Mepazine 增强细胞凋亡并影响细胞活力。 | |||
T68994 | Mepazine hydrochloride monohydrate | ||
Mepazine hydrochloride monohydrate is a MALT1 inhibitor. | |||
T69634 | Mepazine acetate | ||
Mepazine acetate is a MALT1 inhibitor. | |||
T61153 |
Mepazine hydrochloride
|
||
Mepazine hydrochloride (Pecazine hydrochloride) is a potent and selective inhibitor of the MALT1 protease, with IC50 values of 0.83 μM for GSTMALT1 full length and 0.42 μM for GSTMALT1 325-760. It enhances apoptosis and influences the viability of ABC-DLBCL cells [1]. |