Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN1904 |
Magnolignan C
厚朴木酚素C |
Others | Others |
Magnolignan C is a natural product from Magnolia officinalis. | |||
TN1903 |
Magnolignan A
厚朴木脂素A |
Others | Others |
Magnolignan A-2-O-beta-D-glucopyranoside has medium cytotoxic activity against HEp-2 and HepG2 cells, with IC(50) of 13.3 microM, and 46.4 microM, respectively. | |||
TN2268 |
Tetrahydromagnolol
|
Cannabinoid Receptor; GPR; GABA Receptor | Endocrinology/Hormones; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience |
Tetrahydromagnolol 是 Magnolol 的主要代谢产物,是一种弱的GPR55受体拮抗剂。它是选择性大麻素CB2受体激动剂,EC50为 170 nM,Ki 为 416 nM,对CB2受体的选择性比 CB1 受体高 20 倍。 |