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Cat. No. | Product Name | Target | Signaling Pathways |
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T16830 | S-MTC | NOS | Immunology/Inflammation |
S-MTC is a selective inhibitor of type I nitric oxide synthase. | |||
T28120 |
MTC420
MTC-420,MTC 420 |
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MTC420 is a anti-tuberculosis agent with acceptable anti-tuberculosis activity (Mtb IC50 =525 nM, Mtb Wayne IC50 = 76 nM and MDR Mtb patient isolates IC50 = 140 nM). | |||
T21505 |
Suberoyl bis-hydroxamic acid
SBHA,软木肟酸,Suberohydroxamic acid |
Apoptosis; HDAC | Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair |
Suberoyl bis-hydroxamic acid (SBHA) 是一种竞争性且可透过细胞的HDAC1和HDAC3抑制剂,ID50值分别为 0.25 μM 和 0.30 μM。它使肿瘤细胞易于凋亡并促进线粒体凋亡途径,可研究甲状腺髓样癌。 | |||
T38437 |
NMTCA
N-Nitroso-2-methylthiazolidine4-carboxylicacid,NMTPRO,N-nitrosomethylthioproline |
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NMTCA (NMTPRO) is a sulfur-containing N-nitrosamino acid utilized as an endogenous nitrosation indicator in gas chromatography-thermal energy analysis. | |||
T71320 |
ETMTC
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ETMTC is a inhibitor of inflammatory cell adhesion molecules (cams) | |||
T79726 |
RET-IN-25
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RET-IN-25(化合物6b)是一种具有抗癌活性的RET激酶抑制剂。该化合物能够抑制甲状腺髓样癌(MTC),在TT(C634R) MTC细胞系中的IC50值分别为3.6 μM(3天)和3.0 μM(6天)。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T83459 |
11α-O-Tigloyl-12β-O-acetyltenacigenin B
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Aurora Kinase | Cell Cycle/Checkpoint; Chromatin/Epigenetic |
11α-O-Tigloyl-12β-O-acetyltenacigenin B 是Tenacigenin B 的酯类衍生物,源自藤黄藤 (MTC)。该化合物具有调节Aurora-A活性,对淋巴瘤显示出潜在的抗肿瘤效果。 |