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6

抑制剂 & 化合物

1

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Cat. No. Product Name Target Signaling Pathways
T16830 S-MTC

NOS Immunology/Inflammation
S-MTC is a selective inhibitor of type I nitric oxide synthase.
T28120 MTC420

MTC-420,MTC 420

MTC420 is a anti-tuberculosis agent with acceptable anti-tuberculosis activity (Mtb IC50 =525 nM, Mtb Wayne IC50 = 76 nM and MDR Mtb patient isolates IC50 = 140 nM).
T21505 Suberoyl bis-hydroxamic acid

SBHA,软木肟酸,Suberohydroxamic acid

Apoptosis; HDAC Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair
Suberoyl bis-hydroxamic acid (SBHA) 是一种竞争性且可透过细胞的HDAC1和HDAC3抑制剂,ID50值分别为 0.25 μM 和 0.30 μM。它使肿瘤细胞易于凋亡并促进线粒体凋亡途径,可研究甲状腺髓样癌。
T38437 NMTCA

N-Nitroso-2-methylthiazolidine4-carboxylicacid,NMTPRO,N-nitrosomethylthioproline

NMTCA (NMTPRO) is a sulfur-containing N-nitrosamino acid utilized as an endogenous nitrosation indicator in gas chromatography-thermal energy analysis.
T71320 ETMTC

ETMTC is a inhibitor of inflammatory cell adhesion molecules (cams)
T79726 RET-IN-25

RET-IN-25(化合物6b)是一种具有抗癌活性的RET激酶抑制剂。该化合物能够抑制甲状腺髓样癌(MTC),在TT(C634R) MTC细胞系中的IC50值分别为3.6 μM(3天)和3.0 μM(6天)。

化合物

S-MTC
Cat.No: T16830
Synonym:
Target: NOS
MTC420
Cat.No: T28120
Synonym: MTC-420,MTC 420
Target:
Suberoyl bis-hydroxamic acid
Cat.No: T21505
Synonym: SBHA,软木肟酸,Suberohydroxamic acid
Target: Apoptosis, HDAC
NMTCA
Cat.No: T38437
Synonym: N-Nitroso-2-methylthiazolidine4-carboxylicacid,NMTPRO,N-nitrosomethylthioproline
Target:
ETMTC
Cat.No: T71320
Synonym:
Target:
RET-IN-25
Cat.No: T79726
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T83459 11α-O-Tigloyl-12β-O-acetyltenacigenin B

Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic
11α-O-Tigloyl-12β-O-acetyltenacigenin B 是Tenacigenin B 的酯类衍生物,源自藤黄藤 (MTC)。该化合物具有调节Aurora-A活性,对淋巴瘤显示出潜在的抗肿瘤效果。

天然产物

11α-O-Tigloyl-12β-O-acetyltenacigenin B
Cat.No: T83459
Synonym:
Target: Aurora Kinase
TargetMol Loading
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